SCHEMBL8516111

SCHEMBL8516111

O=C(O)N1CCN(S(=O)(=O)c2cc(F)ccc2CBr)CC1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.46
PKM P14618 5/20 0.46
TSHR P16473 1/20 0.43
USP2 O75604 1/20 0.43
GPR183 P32249 2/20 0.41
KDM4E B2RXH2 1/20 0.40
GAA P10253 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
POLB P06746 1/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.40
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
KCNH2 Q12809 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2078886 0.86 ALDH1A1 (0.44) ALDH1A1PKMTSHRUSP2GPR183
SCHEMBL8512706 0.80 TNF (0.54) ALDH1A1PKMTSHRKDM4ESMN1; SMN2
SCHEMBL2082446 0.80 CNR1 (0.50) ALDH1A1PKMTSHRKDM4ESMN1; SMN2
SCHEMBL2077950 0.74 PKM (0.43) ALDH1A1PKMTSHRUSP2GPR183
SCHEMBL29060784 0.71 PKM (0.66) ALDH1A1PKMGPR183GAAL3MBTL1
SCHEMBL12778130 0.70 KDM4E (0.56) ALDH1A1PKMTSHRKDM4EL3MBTL1
SCHEMBL4034882 0.70 TSHR (0.56) ALDH1A1PKMTSHRKDM4EGAA
SCHEMBL2082017 0.69 TSHR (0.49) ALDH1A1PKMTSHRUSP2KDM4E
SCHEMBL14345614 0.69 PKM (0.39) ALDH1A1PKMTSHRUSP2GPR183
SCHEMBL5447251 0.69 ALDH1A1 (0.52) ALDH1A1PKMTSHRGPR183GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2457900-A1 New pyrazole derivatives having CRTh2 antagonistic behaviour Almirall, S.A. (ES) 2012-05-30 EP disclosed