SCHEMBL8513405

SCHEMBL8513405

CN(C)CCN1CCN(c2cccc(-c3ccc4c(c3)C(C)(C)CCC4(C)C)n2)CC1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RARA P10276 2/20 0.45
RARB P10826 2/20 0.45
RAD52 P43351 2/20 0.42
HTR1A P08908 1/20 0.39
DRD2 P14416 1/20 0.39
DRD4 P21917 1/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
HTR7 P34969 1/20 0.39
DRD3 P35462 1/20 0.39
FFAR4 Q5NUL3 1/20 0.37
CFTR P13569 2/20 0.36
KCNH2 Q12809 2/20 0.36
BRD4 O60885 4/20 0.36
CNR1 P21554 2/20 0.36
PIM1 P11309 1/20 0.36
PIM2 Q9P1W9 1/20 0.36
RARG P13631 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12959638 0.87 RARB (0.49) RARARARBRAD52HTR1ADRD2
SCHEMBL8514595 0.85 RARA (0.45) RARARARBRAD52HTR1ADRD2
SCHEMBL31060378 0.85 RARB (0.47) RARARARBRAD52HTR1ADRD2
SCHEMBL8513887 0.85 RARB (0.47) RARARARBRAD52HTR1ADRD2
SCHEMBL12633167 0.84 RARA (0.47) RARARARBHTR1ADRD2DRD4
SCHEMBL12632583 0.84 HTR1A (0.45) RARARARBHTR1ADRD2DRD4
SCHEMBL12959463 0.84 HTR1A (0.45) RARARARBRAD52HTR1ADRD2
SCHEMBL2017413 0.83 RARB (0.54) RARARARBHTR1ADRD2DRD4
SCHEMBL12632929 0.83 RARA (0.46) RARARARBHTR1ADRD2DRD4
SCHEMBL2013393 0.83 RARA (0.46) RARARARBHTR1ADRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO claimed
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed