SCHEMBL8514048

SCHEMBL8514048

CC1(C)CCC(C)(C)c2cc(-c3ccnc(N4CCC5(CCNC5)CC4)n3)ccc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR4 P51679 1/20 0.45
CYP3A4 P08684 2/20 0.42
CYP2D6 P10635 2/20 0.42
TSHR P16473 2/20 0.42
DKK1 O94907 2/20 0.41
ROCK1 Q13464 2/20 0.40
CDC42BPB Q9Y5S2 2/20 0.40
ROCK2 O75116 1/20 0.40
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
HSD17B10 Q99714 1/20 0.38
RARA P10276 1/20 0.38
RARB P10826 1/20 0.38
KCNH2 Q12809 1/20 0.38
HDAC1 Q13547 1/20 0.38
PIK3CA P42336 2/20 0.37
CYP11B1 P15538 1/20 0.37
PIK3CD O00329 1/20 0.37
PIK3R1 P27986 1/20 0.37
PIK3CB P42338 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8511327 0.99 CCR4 (0.46) CCR4CYP3A4CYP2D6TSHRDKK1
SCHEMBL8514182 0.97 CCR4 (0.43) CCR4CYP3A4CYP2D6TSHRDKK1
SCHEMBL8512407 0.87 ADRB1 (0.44) DKK1ROCK2ALDH1A1RARARARB
Hydrochloric Acid SCHEMBL8512430 0.85 ADRB1 (0.43) DKK1ROCK2ALDH1A1RARARARB
SCHEMBL8515840 0.85 ROCK1 (0.41) CCR4CYP3A4CYP2D6TSHRROCK1
SCHEMBL8510102 0.82 PIM1 (0.46) CYP3A4CYP2D6TSHRALDH1A1CYP1A2
Hydrochloric Acid SCHEMBL8513898 0.81 PIM1 (0.46) CYP3A4CYP2D6TSHRALDH1A1CYP1A2
Hydrochloric Acid SCHEMBL8514984 0.81 TBK1 (0.42) CCR4RARARARBKCNH2HDAC1
SCHEMBL8514868 0.80 DKK1 (0.64) DKK1ROCK2RARARARBPIK3CA
Hydrochloric Acid SCHEMBL8511494 0.79 DKK1 (0.63) DKK1ROCK2RARARARBPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO claimed