SCHEMBL8514162

SCHEMBL8514162

CC1(C)CCC(C)(C)c2cc(-c3cc(N4CCC(N)CC4)ccn3)ccc21.CC1(C)CCC(C)(C)c2cc(-c3cc(N4CCC5(CCNC5)CC4)ccn3)ccc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 3/20 0.38
CDC42BPB Q9Y5S2 3/20 0.38
ROCK2 O75116 2/20 0.38
HDAC1 Q13547 5/20 0.37
KCNH2 Q12809 4/20 0.37
DKK1 O94907 1/20 0.36
USP2 O75604 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TP53 P04637 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
HSD17B10 Q99714 1/20 0.35
HRH4 Q9H3N8 3/20 0.35
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
PIM1 P11309 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8515840 0.93 ROCK1 (0.41) ROCK1CDC42BPBROCK2HDAC1KCNH2
SCHEMBL8510961 0.89 DKK1 (0.43) HDAC1DKK1HRH4PIM1RARA
Trifluoroacetic Acid SCHEMBL8511708 0.85 HDAC1 (0.39) ROCK1CDC42BPBROCK2HDAC1KCNH2
SCHEMBL9612706 0.80 HTR7 (0.49) HRH4PIM1
SCHEMBL8514048 0.79 CCR4 (0.45) ROCK1CDC42BPBROCK2HDAC1KCNH2
Hydrochloric Acid SCHEMBL8511327 0.78 CCR4 (0.46) ROCK1CDC42BPBROCK2HDAC1KCNH2
SCHEMBL8514182 0.77 CCR4 (0.43) ROCK1CDC42BPBROCK2HDAC1KCNH2
SCHEMBL8515164 0.74 HRH4 (0.43) HDAC1HRH4RARARARBRARG
SCHEMBL8514439 0.74 LRRK2 (0.45) ALDH1A1CYP1A2HSD17B10HRH4
SCHEMBL8514868 0.74 DKK1 (0.64) ROCK2DKK1RARARARBHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO claimed