SCHEMBL8514728

SCHEMBL8514728

CC(C)Oc1ccc(-c2nccc(N3CCC(NC(=O)O)CC3)n2)cc1C(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 2/20 0.41
HMOX1 P09601 1/20 0.41
USP2 O75604 1/20 0.39
HPGD P15428 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ACACB O00763 1/20 0.39
ALDH1A1 P00352 1/20 0.38
TSHR P16473 1/20 0.38
CETP P11597 3/20 0.37
HRH4 Q9H3N8 1/20 0.37
KIT P10721 1/20 0.37
MAPK14 Q16539 1/20 0.37
CKS1B P61024 2/20 0.37
SKP1 P63208 2/20 0.37
SKP2 Q13309 2/20 0.37
S1PR1 P21453 1/20 0.36
PIK3CD O00329 1/20 0.36
PIK3CA P42336 1/20 0.36
KCNH2 Q12809 1/20 0.36
GSK3B P49841 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8515012 0.93 XDH (0.39) XDHHMOX1USP2HPGDSMN1; SMN2
SCHEMBL8511963 0.84 HRH3 (0.45) XDHUSP2ACACBALDH1A1TSHR
Hydrochloric Acid SCHEMBL8511187 0.83 HRH3 (0.44) XDHUSP2ACACBALDH1A1TSHR
SCHEMBL8511517 0.80 CYP1A2 (0.40) XDHUSP2ALDH1A1TSHRPIK3CD
SCHEMBL8514719 0.76 HRH3 (0.45) XDHUSP2ACACBALDH1A1TSHR
SCHEMBL8515197 0.76 RARB (0.42) USP2HPGDSMN1; SMN2ACACBALDH1A1
Hydrochloric Acid SCHEMBL8514774 0.75 HRH3 (0.44) XDHUSP2ACACBALDH1A1TSHR
SCHEMBL8515116 0.73 CYP1A2 (0.40) XDHUSP2ALDH1A1TSHRPIK3CD
SCHEMBL8514151 0.72 CYP1A2 (0.40) XDHUSP2ALDH1A1TSHRPIK3CD
SCHEMBL4334757 0.69 TRPV1 (0.51) CKS1BSKP1SKP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed