SCHEMBL8511517

SCHEMBL8511517

CC(C)Oc1ccc(-c2nccc(N3CC[CH]CC3)n2)cc1C(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 5/20 0.40
ALDH1A1 P00352 4/20 0.40
CYP3A4 P08684 4/20 0.40
HSD17B10 Q99714 3/20 0.40
CLK4 Q9HAZ1 2/20 0.40
USP2 O75604 2/20 0.40
CASP1 P29466 1/20 0.40
CASP7 P55210 1/20 0.40
XDH P47989 1/20 0.39
PIK3CD O00329 2/20 0.38
PIK3CA P42336 2/20 0.38
CYP2D6 P10635 3/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.37
CYP2C19 P33261 2/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ATR Q13535 10/20 0.35
ATRIP Q8WXE1 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8514151 0.91 CYP1A2 (0.40) CYP1A2ALDH1A1CYP3A4HSD17B10CLK4
SCHEMBL8511963 0.86 HRH3 (0.45) CYP1A2ALDH1A1CYP3A4HSD17B10CLK4
Hydrochloric Acid SCHEMBL8511187 0.85 HRH3 (0.44) CYP1A2ALDH1A1CYP3A4HSD17B10CLK4
SCHEMBL8515116 0.81 CYP1A2 (0.40) CYP1A2ALDH1A1CYP3A4HSD17B10CLK4
SCHEMBL8514728 0.80 XDH (0.41) ALDH1A1USP2XDHPIK3CDPIK3CA
SCHEMBL8514640 0.79 ITGB2 (0.41) CYP1A2ALDH1A1HSD17B10TSHRKDM4E
SCHEMBL8514719 0.78 HRH3 (0.45) CYP1A2ALDH1A1CYP3A4HSD17B10CLK4
Hydrochloric Acid SCHEMBL8514774 0.77 HRH3 (0.44) CYP1A2ALDH1A1CYP3A4HSD17B10CLK4
SCHEMBL8515012 0.72 XDH (0.39) CYP1A2ALDH1A1CYP3A4USP2XDH
SCHEMBL8513449 0.70 S1PR1 (0.42) CYP1A2ALDH1A1CYP3A4HSD17B10CLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed