SCHEMBL8514719

SCHEMBL8514719

CC(C)Oc1cc(-c2nccc(N3CCC(N)CC3)n2)ccc1C(C)C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.45
DKK1 O94907 1/20 0.38
CYP1A2 P05177 5/20 0.38
ALDH1A1 P00352 3/20 0.38
HSD17B10 Q99714 3/20 0.38
CYP3A4 P08684 3/20 0.38
CLK4 Q9HAZ1 2/20 0.38
USP2 O75604 1/20 0.38
CASP1 P29466 1/20 0.38
CASP7 P55210 1/20 0.38
PDE4D Q08499 1/20 0.37
PIK3CD O00329 1/20 0.36
PIK3CA P42336 1/20 0.36
CYP2D6 P10635 3/20 0.36
ALOX15 P16050 2/20 0.36
HRH4 Q9H3N8 4/20 0.35
TSHR P16473 2/20 0.35
ACACB O00763 1/20 0.35
XDH P47989 1/20 0.35
ATR Q13535 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8514774 0.99 HRH3 (0.44) HRH3DKK1CYP1A2ALDH1A1HSD17B10
SCHEMBL8511963 0.92 HRH3 (0.45) HRH3DKK1CYP1A2ALDH1A1HSD17B10
Hydrochloric Acid SCHEMBL8511187 0.91 HRH3 (0.44) HRH3DKK1CYP1A2ALDH1A1HSD17B10
SCHEMBL8515116 0.87 CYP1A2 (0.40) CYP1A2ALDH1A1HSD17B10CYP3A4CLK4
SCHEMBL8514151 0.86 CYP1A2 (0.40) CYP1A2ALDH1A1HSD17B10CYP3A4CLK4
SCHEMBL8515012 0.84 XDH (0.39) CYP1A2ALDH1A1CYP3A4USP2PIK3CD
SCHEMBL8511517 0.78 CYP1A2 (0.40) CYP1A2ALDH1A1HSD17B10CYP3A4CLK4
SCHEMBL8514728 0.76 XDH (0.41) ALDH1A1USP2PIK3CDPIK3CAHRH4
SCHEMBL8511419 0.72 KARS1 (0.37) CYP1A2HSD17B10HRH4KARS1
SCHEMBL2049616 0.72 HRH3 (0.49) HRH3DKK1CYP1A2ALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO claimed
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed