SCHEMBL8514830

SCHEMBL8514830

CC1(C)CCC(C)(C)c2cc(-c3cc(-c4ccc(C5(N)CCC5)cc4)ccn3)ccc21

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
RARA P10276 8/20 0.40
RARB P10826 7/20 0.40
RARG P13631 6/20 0.40
AKT1 P31749 9/20 0.39
AKT2 P31751 4/20 0.39
RXRA P19793 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8513591 0.96 RARA (0.38) RARARARBRARGAKT1AKT2
Hydrochloric Acid SCHEMBL8510905 0.95 RARA (0.38) RARARARBRARGAKT1AKT2
Trifluoroacetic Acid SCHEMBL8511940 0.89 RARB (0.42) RARARARBRARGAKT1RXRA
SCHEMBL18961191 0.85 RARA (0.47) RARARARBRARGRXRA
SCHEMBL8511696 0.84 RARB (0.44) RARARARBRARGAKT1AKT2
Hydrochloric Acid SCHEMBL8515237 0.83 RARB (0.44) RARARARBRARGAKT1AKT2
SCHEMBL16998655 0.82 RARB (0.49) RARARARBRARGRXRA
SCHEMBL16998862 0.81 RARB (0.55) RARARARBRARGRXRA
SCHEMBL8515374 0.80 RARB (0.60) RARARARBRARGAKT1AKT2
Hydrochloric Acid SCHEMBL8612658 0.79 RARA (0.58) RARARARBRARGAKT1AKT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO claimed
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed