SCHEMBL8515192

SCHEMBL8515192

CC(C)(C)OC(=O)N1CCC2(CCN(c3cccc(-c4ccc5c(c4)C(C)(C)CCC5(C)C)n3)CC2)C1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 1/20 0.50
RARA P10276 1/20 0.46
RARB P10826 1/20 0.46
SCD5 Q86SK9 1/20 0.44
HDAC2 Q92769 2/20 0.44
RET P07949 5/20 0.42
ACACB O00763 5/20 0.41
HDAC1 Q13547 1/20 0.40
KIF18A Q8NI77 1/20 0.40
USP30 Q70CQ3 1/20 0.39
RORC P51449 1/20 0.39
GPR119 Q8TDV5 1/20 0.38
CKS1B P61024 1/20 0.38
SKP1 P63208 1/20 0.38
SKP2 Q13309 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2015994 0.90 RARA (0.50) RARARARBRETKIF18AGPR119
SCHEMBL12804321 0.86 CKS1B (0.51) RARARARBRETKIF18AGPR119
SCHEMBL8514114 0.85 CYP11B2 (0.47) CYP11B2SCD5HDAC2RETACACB
SCHEMBL2016042 0.84 CKS1B (0.48) RARARARBRETKIF18AGPR119
SCHEMBL12633005 0.83 RARA (0.44) RARARARBKIF18AGPR119CKS1B
SCHEMBL8511358 0.83 CYP11B2 (0.46) CYP11B2SCD5HDAC2RETACACB
SCHEMBL2016854 0.81 CKS1B (0.45) RARARARBRETKIF18AGPR119
SCHEMBL12633907 0.80 CKS1B (0.46) RARARARBRETKIF18AGPR119
Hydrochloric Acid SCHEMBL8514984 0.80 TBK1 (0.42) RARARARBHDAC1KIF18AGPR119
SCHEMBL2015302 0.79 CKS1B (0.43) RARARARBRETKIF18AUSP30

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed