SCHEMBL8515262

SCHEMBL8515262

CC1(C)CCC(C)(C)c2cc(-c3cccc(N4CCC(NC(=N)N)CC4)n3)ccc21

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RARA P10276 2/20 0.45
RARB P10826 2/20 0.45
CCNT1 O60563 4/20 0.40
CNR1 P21554 7/20 0.38
RARG P13631 2/20 0.37
PIM1 P11309 1/20 0.36
PIM3 Q86V86 1/20 0.36
PIM2 Q9P1W9 1/20 0.36
SMO Q99835 1/20 0.36
KARS1 Q15046 2/20 0.36
BTK Q06187 1/20 0.35
HSD11B1 P28845 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8612509 0.99 RARA (0.44) RARARARBCCNT1CNR1RARG
SCHEMBL12632945 0.84 RARB (0.56) RARARARBCCNT1CNR1RARG
SCHEMBL8510951 0.83 DKK1 (0.45) RARARARBSMO
SCHEMBL12633193 0.83 RARA (0.45) RARARARBCCNT1CNR1RARG
SCHEMBL8515149 0.83 RARA (0.49) RARARARBPIM1PIM3PIM2
SCHEMBL12633266 0.82 RARB (0.45) RARARARBCCNT1CNR1RARG
Hydrochloric Acid SCHEMBL8512387 0.82 DKK1 (0.44) RARARARBSMO
SCHEMBL12632966 0.82 RARB (0.45) RARARARBCCNT1CNR1RARG
Hydrochloric Acid SCHEMBL8515557 0.82 RARA (0.48) RARARARBPIM1PIM3PIM2
Hydrochloric Acid SCHEMBL2015173 0.82 RARA (0.48) RARARARBPIM1PIM3PIM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO claimed
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed