SCHEMBL8515328

SCHEMBL8515328

C(#Cc1cccc(-c2ncc3ccccc3n2)n1)c1ccccn1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 7/20 0.59
KCNH2 Q12809 2/20 0.59
CYP1A2 P05177 5/20 0.42
METAP1 P53582 2/20 0.36
KDM4E B2RXH2 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
LMNA P02545 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
TP53 P04637 1/20 0.36
ALPL P05186 1/20 0.36
HSP90AA1 P07900 1/20 0.36
ALPI P09923 1/20 0.36
ALPG P10696 1/20 0.36
ALOX15 P16050 1/20 0.36
MAPK1 P28482 1/20 0.36
CCR1 P32246 1/20 0.36
HTT P42858 1/20 0.36
CCR5 P51681 1/20 0.36
CCR8 P51685 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8778633 0.86 GRM5 (0.46) GRM5KCNH2CYP1A2KDM4ELMNA
SCHEMBL8778606 0.81 CYP1A2 (0.42) GRM5KCNH2CYP1A2KDM4ELMNA
SCHEMBL45359 0.80 KDM4E (0.57) CYP1A2METAP1KDM4ETDP1LMNA
SCHEMBL29784044 0.80 KDM4E (0.57) CYP1A2METAP1KDM4ETDP1LMNA
SCHEMBL8778608 0.80 CYP1A2 (0.40) GRM5KCNH2CYP1A2
SCHEMBL8778641 0.78 GRM5 (0.40) GRM5KCNH2CYP1A2
SCHEMBL15877252 0.75 GRM5 (1.00) GRM5KCNH2CYP1A2KDM4ESMN1; SMN2
SCHEMBL8515946 0.74 KDM4E (0.43) GRM5CYP1A2METAP1KDM4ETDP1
SCHEMBL3784385 0.72 RAB9A (0.55) CYP1A2LMNASMN1; SMN2NPC1RAB9A
SCHEMBL3788203 0.72 CYP1A2 (0.45) CYP1A2METAP1KDM4ETDP1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069601-A1 SUBSTITUTED QUINAZOLINES AS FUNGICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-05-31 WO disclosed