SCHEMBL8515822

SCHEMBL8515822

CC(C)(C)c1cc(-c2nccc(N3CCNCC3)n2)ccc1NC1CCCC1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PRKD1 Q15139 14/20 0.46
PRKD2 Q9BZL6 7/20 0.46
ADRB1 P08588 1/20 0.45
CYP1A2 P05177 2/20 0.43
CYP2C9 P11712 1/20 0.43
HSD17B10 Q99714 1/20 0.43
HRH4 Q9H3N8 4/20 0.43
HRH3 Q9Y5N1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8511658 0.83 GPR119 (0.46) PRKD1PRKD2HRH4
SCHEMBL8515459 0.82 PRKD1 (0.46) PRKD1PRKD2ADRB1
SCHEMBL1588027 0.72 HRH4 (0.71) PRKD1PRKD2HRH4HRH3
SCHEMBL1588677 0.67 HRH4 (0.67) HRH4HRH3
SCHEMBL8515571 0.67 CYP1A2 (0.47) PRKD1PRKD2ADRB1CYP1A2CYP2C9
SCHEMBL1579219 0.67 PRKD1 (0.71) PRKD1PRKD2ADRB1
SCHEMBL8515830 0.67 PRKD1 (0.45) PRKD1PRKD2ADRB1
Hydrochloric Acid SCHEMBL8514610 0.66 CYP1A2 (0.46) PRKD1PRKD2ADRB1CYP1A2CYP2C9
SCHEMBL1579273 0.66 PRKD1 (0.79) PRKD1PRKD2ADRB1
SCHEMBL3272539 0.66 PIK3CD (0.52) ADRB1CYP1A2CYP2C9HSD17B10HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO claimed
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed