SCHEMBL8515949

SCHEMBL8515949

CCOC(=O)CC(=O)c1ccc(Cc2ccc(OC(F)(F)F)cc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.56
EPHX2 P34913 5/20 0.53
PPARG P37231 2/20 0.53
PPARA Q07869 2/20 0.53
HDAC3 O15379 4/20 0.48
HDAC1 Q13547 4/20 0.48
HDAC2 Q92769 4/20 0.48
HDAC4 P56524 3/20 0.47
HDAC7 Q8WUI4 3/20 0.47
HDAC10 Q969S8 3/20 0.47
HDAC11 Q96DB2 3/20 0.47
HDAC8 Q9BY41 3/20 0.47
HDAC6 Q9UBN7 3/20 0.47
HDAC9 Q9UKV0 3/20 0.47
HDAC5 Q9UQL6 3/20 0.47
OPRK1 P41145 1/20 0.47
NR1H4 Q96RI1 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5100087 0.93 POLB (0.63) POLBEPHX2PPARGPPARAHDAC3
SCHEMBL9607170 0.83 RAB9A (0.51) EPHX2PPARGPPARAHDAC3HDAC1
SCHEMBL8514914 0.82 SMN1; SMN2 (0.50) SMN1; SMN2NPC1RAB9AHPGDMAPT
SCHEMBL27809101 0.81 POLB (0.62) POLBEPHX2PPARGPPARAHDAC3
SCHEMBL17290763 0.80 HDAC3 (0.52) POLBEPHX2HDAC3HDAC1HDAC2
SCHEMBL4994157 0.80 ALDH1A1 (0.51) POLBSMN1; SMN2NPC1RAB9AHPGD
SCHEMBL20351685 0.80 POLB (0.60) POLBEPHX2PPARGPPARAHDAC3
SCHEMBL508864 0.79 MRGPRX4 (0.57) EPHX2HDAC3HDAC1HDAC2HDAC4
SCHEMBL1940297 0.79 POLB (0.62) POLBEPHX2PPARGPPARAHDAC4
SCHEMBL2743506 0.78 POLB (0.56) POLBEPHX2PPARGPPARAHDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed