SCHEMBL851679

SCHEMBL851679

N#Cc1ccc(COc2cc(Oc3cccc(C(=O)O)c3)ccc2C#N)cc1

nearest known ligand 0.60

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SMPD1 P17405 1/20 0.54
MRGPRX4 Q96LA9 7/20 0.54
NR4A2 P43354 4/20 0.51
PTGER1 P34995 3/20 0.48
XDH P47989 1/20 0.47
NR4A1 P22736 1/20 0.47
NR4A3 Q92570 1/20 0.47
CYP11B1 P15538 1/20 0.47
CYP11B2 P19099 1/20 0.47
AKR1C3 P42330 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL851731 0.90 MRGPRX4 (0.58) MRGPRX4NR4A2
SCHEMBL25214512 0.83 SMPD1 (0.74) SMPD1MRGPRX4NR4A2NR4A1NR4A3
SCHEMBL30392119 0.83 SMPD1 (0.74) SMPD1MRGPRX4NR4A2NR4A1NR4A3
SCHEMBL13268612 0.80 AKR1C3 (0.72) AKR1C3
SCHEMBL851693 0.80 MRGPRX4 (0.46) MRGPRX4NR4A2XDHNR4A1NR4A3
SCHEMBL4684138 0.78 MRGPRX4 (0.70) MRGPRX4NR4A2
SCHEMBL27875417 0.76 AKR1C3 (0.65) MRGPRX4AKR1C3
SCHEMBL851678 0.76 MEN1 (0.60) SMPD1MRGPRX4NR4A2NR4A1NR4A3
SCHEMBL851559 0.76 MRGPRX4 (0.49) MRGPRX4NR4A2NR4A1NR4A3
SCHEMBL851770 0.75 AKR1C3 (0.52) SMPD1MRGPRX4NR4A2AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2432556-A1 PROTEASE INHIBITORS Orion Corporation (FI) 2012-03-28 EP disclosed
WO-2010133748-A1 PROTEASE INHIBITORS ORION CORPORATION (FI) 2010-11-25 WO disclosed