SCHEMBL851693

SCHEMBL851693

CC(C)(C)OC(=O)C(N)c1ccc(COc2cc(Oc3cccc(C(=O)O)c3)ccc2C#N)cc1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 9/20 0.46
NR4A2 P43354 4/20 0.45
NR4A1 P22736 1/20 0.45
NR4A3 Q92570 1/20 0.45
XDH P47989 3/20 0.41
NPC1 O15118 1/20 0.40
POLB P06746 1/20 0.40
CYP2C9 P11712 1/20 0.40
RAB9A P51151 1/20 0.40
FFAR1 O14842 1/20 0.38
FFAR4 Q5NUL3 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL851559 0.92 MRGPRX4 (0.49) MRGPRX4NR4A2NR4A1NR4A3NPC1
SCHEMBL851679 0.80 SMPD1 (0.54) MRGPRX4NR4A2NR4A1NR4A3XDH
SCHEMBL851694 0.79 RAB9A (0.44) MRGPRX4NR4A2NR4A1NR4A3NPC1
SCHEMBL851731 0.76 MRGPRX4 (0.58) MRGPRX4NR4A2RAB9AFFAR1FFAR4
SCHEMBL851560 0.73 MRGPRX4 (0.43) MRGPRX4NR4A2RAB9AFFAR1FFAR4
SCHEMBL852056 0.72 PARP15 (0.44) NPC1POLBCYP2C9RAB9AFFAR1
SCHEMBL851237 0.71 RAB9A (0.44) NPC1RAB9AFFAR1
SCHEMBL184424 0.70 ANPEP (0.51) NR4A2NR4A1NR4A3
SCHEMBL2570186 0.69 LMNA (0.49) NPC1RAB9A
SCHEMBL27875417 0.67 AKR1C3 (0.65) MRGPRX4NPC1POLBCYP2C9RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2432556-A1 PROTEASE INHIBITORS Orion Corporation (FI) 2012-03-28 EP disclosed
WO-2010133748-A1 PROTEASE INHIBITORS ORION CORPORATION (FI) 2010-11-25 WO disclosed