SCHEMBL8517468

SCHEMBL8517468

C=CCOc1cnc(-c2ccccc2C#CC(C)O)nc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.39
MAPT P10636 2/20 0.39
ADRB2 P07550 4/20 0.38
ADRB1 P08588 4/20 0.38
LMNA P02545 2/20 0.38
SLC22A1 O15245 1/20 0.38
CYP1A2 P05177 1/20 0.38
HTR1A P08908 1/20 0.38
HTR2A P28223 1/20 0.38
SLC6A4 P31645 1/20 0.38
ADRA1A P35348 1/20 0.38
ACACB O00763 1/20 0.36
ADRB3 P13945 3/20 0.36
ALDH1A1 P00352 1/20 0.35
PTPRC P08575 1/20 0.34
CHRNB2 P17787 3/20 0.34
CHRNB4 P30926 3/20 0.34
CHRNA3 P32297 3/20 0.34
CHRNA4 P43681 3/20 0.34
ATM Q13315 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8517770 0.84 ADRB2 (0.32) CYP2D6ADRB2ADRB1LMNACYP1A2
SCHEMBL8517467 0.81 LMNA (0.40) CYP2D6MAPTADRB2ADRB1LMNA
SCHEMBL7856830 0.80 MAPT (0.41) CYP2D6MAPTADRB2ADRB1LMNA
SCHEMBL8517374 0.80 ADRB2 (0.44) CYP2D6MAPTADRB2ADRB1LMNA
SCHEMBL8518542 0.77 ADRB2 (0.35) CYP2D6MAPTADRB2ADRB1LMNA
SCHEMBL8517691 0.72 ADRB2 (0.44) CYP2D6MAPTADRB2ADRB1LMNA
SCHEMBL8518534 0.72 LMNA (0.37) CYP2D6MAPTADRB2ADRB1LMNA
SCHEMBL8517500 0.72 ADRB2 (0.39) CYP2D6ADRB2ADRB1LMNACYP1A2
SCHEMBL8517707 0.70 CYP2D6 (0.51) CYP2D6MAPTADRB2ADRB1LMNA
SCHEMBL7863562 0.69 ADRB2 (0.46) CYP2D6MAPTADRB2ADRB1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628530-B1 ACETYLENE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, LIQUID CRYSTAL COMPOSITION CONTAINING THE SAME AS ACTIVE INGREDIENT, AND LIQUID CRYSTAL ELEMENT MADE THEREFROM SUMITOMO CHEMICAL CO (JP) 1999-03-24 EP disclosed
US-5534188-A Acetylene derivatives, process for producing the same, liquid crystal composition containing the same as an active ingredient, and liquid crystal element using said liquid crystal composition SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1996-07-09 US disclosed
EP-0628530-A1 ACETYLENE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, LIQUID CRYSTAL COMPOSITION CONTAINING THE SAME AS ACTIVE INGREDIENT, AND LIQUID CRYSTAL ELEMENT MADE THEREFROM SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1994-12-14 EP disclosed