SCHEMBL8518534

SCHEMBL8518534

C=CCOc1ccc(C#CC(C)O)c(-c2cccnn2)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.37
MEN1 O00255 1/20 0.37
MAPT P10636 1/20 0.37
KMT2A Q03164 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CYP2D6 P10635 2/20 0.37
ADRB2 P07550 3/20 0.34
ADRB1 P08588 3/20 0.34
ADRB3 P13945 2/20 0.34
MAOA P21397 1/20 0.32
ALDH1A1 P00352 2/20 0.31
SLC22A1 O15245 1/20 0.31
CYP1A2 P05177 1/20 0.31
HTR1A P08908 1/20 0.31
HTR2A P28223 1/20 0.31
SLC6A4 P31645 1/20 0.31
ADRA1A P35348 1/20 0.31
FGFR1 P11362 1/20 0.31
ACACB O00763 1/20 0.30
CHRNB2 P17787 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8517467 0.84 LMNA (0.40) LMNAMEN1MAPTKMT2ASMN1; SMN2
SCHEMBL8517829 0.82 GABRA1 (0.36) LMNAMEN1MAPTKMT2ASMN1; SMN2
SCHEMBL8518542 0.73 ADRB2 (0.35) LMNAMAPTCYP2D6ADRB2ADRB1
SCHEMBL8517468 0.72 CYP2D6 (0.39) LMNAMEN1MAPTKMT2ASMN1; SMN2
SCHEMBL8517137 0.69 CYP2D6 (0.48) LMNAMEN1MAPTKMT2ASMN1; SMN2
SCHEMBL8517692 0.67 ADRB2 (0.39) MEN1KMT2ACYP2D6ADRB2ADRB1
SCHEMBL8517707 0.67 CYP2D6 (0.51) LMNAMEN1MAPTKMT2ASMN1; SMN2
SCHEMBL8517135 0.67 CYP2D6 (0.43) LMNAMAPTSMN1; SMN2CYP2D6ADRB2
SCHEMBL8601719 0.66 DCTPP1 (0.33) DCTPP1MGAMGAASIMGAM2
SCHEMBL8517666 0.66 CYP2D6 (0.40) LMNAMEN1MAPTKMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628530-B1 ACETYLENE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, LIQUID CRYSTAL COMPOSITION CONTAINING THE SAME AS ACTIVE INGREDIENT, AND LIQUID CRYSTAL ELEMENT MADE THEREFROM SUMITOMO CHEMICAL CO (JP) 1999-03-24 EP disclosed
US-5534188-A Acetylene derivatives, process for producing the same, liquid crystal composition containing the same as an active ingredient, and liquid crystal element using said liquid crystal composition SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1996-07-09 US disclosed
EP-0628530-A1 ACETYLENE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, LIQUID CRYSTAL COMPOSITION CONTAINING THE SAME AS ACTIVE INGREDIENT, AND LIQUID CRYSTAL ELEMENT MADE THEREFROM SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1994-12-14 EP disclosed