SCHEMBL8517630

SCHEMBL8517630

C=CCOc1nccnc1-c1cccc(C#CC(C)O)c1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.34
ADRB2 P07550 2/20 0.33
ADRB1 P08588 2/20 0.33
SLC22A1 O15245 1/20 0.33
LMNA P02545 1/20 0.33
CYP1A2 P05177 1/20 0.33
HTR1A P08908 1/20 0.33
HTR2A P28223 1/20 0.33
SLC6A4 P31645 1/20 0.33
ADRA1A P35348 1/20 0.33
MAPT P10636 1/20 0.32
ADRB3 P13945 1/20 0.32
FGFR3 P22607 1/20 0.31
KDR P35968 1/20 0.31
BACE1 P56817 1/20 0.30
SQOR Q9Y6N5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8517724 0.82 FGFR3 (0.32) FGFR3KDR
SCHEMBL8517606 0.78 ASIC3 (0.35) CYP2D6ADRB2ADRB1SLC22A1LMNA
SCHEMBL8517940 0.71 ASIC3 (0.36) FGFR3KDR
SCHEMBL8517605 0.70 ADRB2 (0.39) CYP2D6ADRB2ADRB1SLC22A1LMNA
SCHEMBL8517707 0.69 CYP2D6 (0.51) CYP2D6ADRB2ADRB1SLC22A1LMNA
SCHEMBL8517137 0.69 CYP2D6 (0.48) CYP2D6ADRB2ADRB1LMNAMAPT
SCHEMBL8670095 0.68 CASR (0.33) CYP2D6BACE1
SCHEMBL8517692 0.67 ADRB2 (0.39) CYP2D6ADRB2ADRB1ADRB3
SCHEMBL8517627 0.67 CYP2D6 (0.34) CYP2D6ADRB2ADRB1SLC22A1LMNA
SCHEMBL8517269 0.66 CYP2D6 (0.35) CYP2D6ADRB2ADRB1SLC22A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628530-B1 ACETYLENE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, LIQUID CRYSTAL COMPOSITION CONTAINING THE SAME AS ACTIVE INGREDIENT, AND LIQUID CRYSTAL ELEMENT MADE THEREFROM SUMITOMO CHEMICAL CO (JP) 1999-03-24 EP disclosed
US-5534188-A Acetylene derivatives, process for producing the same, liquid crystal composition containing the same as an active ingredient, and liquid crystal element using said liquid crystal composition SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1996-07-09 US disclosed
EP-0628530-A1 ACETYLENE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, LIQUID CRYSTAL COMPOSITION CONTAINING THE SAME AS ACTIVE INGREDIENT, AND LIQUID CRYSTAL ELEMENT MADE THEREFROM SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1994-12-14 EP disclosed