Guanidine

Guanidine

SCHEMBL8518148

CC(=Cc1ccc(Oc2cccnc2)c(C(F)(F)F)c1)C(=O)O.Cl.Cl.N=C(N)N

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

KCNA1KCNA10KCNA2KCNA3KCNA4KCNA5KCNA6KCNA7KCNB1KCNB2KCNC1KCNC2KCNC3KCNC4KCND1KCND2KCND3KCNF1KCNG1KCNG2KCNG3KCNG4KCNH1KCNH2KCNH3KCNH4KCNH5KCNH6KCNH7KCNH8KCNQ1KCNQ2KCNQ3KCNQ4KCNQ5KCNS1KCNS2KCNS3KCNV1KCNV2

The experimentally established mechanism targets of Guanidine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.46
TBXAS1 P24557 6/20 0.44
SUCNR1 Q9BXA5 1/20 0.38
ALDH1A1 P00352 2/20 0.38
CYP1A2 P05177 1/20 0.37
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
HTR2B P41595 1/20 0.37
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
GAA P10253 1/20 0.36
MAPK1 P28482 1/20 0.36
KMT2A Q03164 1/20 0.36
RECQL P46063 1/20 0.36
HIF1A Q16665 1/20 0.36
EGFR P00533 1/20 0.36
PDGFRB P09619 1/20 0.36
PDGFRA P16234 1/20 0.36
SCN9A Q15858 1/20 0.35
CFTR P13569 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8438436 0.95 TBXAS1 (0.46) SMN1; SMN2TBXAS1SUCNR1ALDH1A1CYP1A2
SCHEMBL8374897 0.95 TBXAS1 (0.46) SMN1; SMN2TBXAS1SUCNR1ALDH1A1CYP1A2
SCHEMBL8374491 0.82 MEN1 (0.46) SMN1; SMN2TBXAS1SUCNR1ALDH1A1CYP1A2
SCHEMBL8374493 0.82 MEN1 (0.46) SMN1; SMN2TBXAS1SUCNR1ALDH1A1CYP1A2
Hydrochloric Acid SCHEMBL10982425 0.76 TBXAS1 (0.61) TBXAS1ALDH1A1GAARECQL
Hydrochloric Acid SCHEMBL10992507 0.76 TBXAS1 (0.61) TBXAS1ALDH1A1GAARECQL
Hydrochloric Acid SCHEMBL8379790 0.75 SMN1; SMN2 (0.48) SMN1; SMN2ALDH1A1CYP1A2HTR2AHTR2C
SCHEMBL10987986 0.75 TBXAS1 (0.59) TBXAS1ALDH1A1GAARECQL
SCHEMBL10987989 0.75 TBXAS1 (0.59) TBXAS1ALDH1A1GAARECQL
SCHEMBL8831863 0.73 SMN1; SMN2 (0.49) SMN1; SMN2ALDH1A1KDM4EMEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5883133-A CARDIOVASCULAR DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1999-03-16 US disclosed