SCHEMBL8518362

SCHEMBL8518362

O=C(Nc1ccc2c(c1)OC(F)(F)O2)C(F)(F)F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
USP36 Q9P275 1/20 0.47
SMN1; SMN2 Q16637 3/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
RECQL P46063 1/20 0.46
ADORA3 P0DMS8 1/20 0.45
ADORA2A P29274 1/20 0.45
ADORA2B P29275 1/20 0.45
ADORA1 P30542 1/20 0.45
BRAF P15056 1/20 0.45
GAA P10253 1/20 0.44
ALDH1A1 P00352 5/20 0.44
MAPT P10636 3/20 0.44
NPSR1 Q6W5P4 1/20 0.44
KIF11 P52732 1/20 0.43
KDM4E B2RXH2 3/20 0.43
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26633294 0.82 ADORA3 (0.51) CYP1A2CYP2C9CYP2C19USP36SMN1; SMN2
SCHEMBL15553344 0.81 BRAF (0.58) CYP1A2CYP2C9CYP2C19SMN1; SMN2RECQL
SCHEMBL4053608 0.80 EPHX2 (0.61) CYP1A2CYP2C9CYP2C19USP36SMN1; SMN2
SCHEMBL19678085 0.77 KIT (0.56) SMN1; SMN2BRAFALDH1A1MAPTNPSR1
SCHEMBL22648397 0.77 RECQL (0.54) CYP1A2SMN1; SMN2RECQLADORA3ADORA2A
SCHEMBL4053993 0.76 MAPT (0.62) CYP1A2CYP2C9CYP2C19SMN1; SMN2BRAF
SCHEMBL4057629 0.76 NPC1 (0.61) SMN1; SMN2ADORA3ALDH1A1MAPT
SCHEMBL19668020 0.76 RAB9A (0.51) SMN1; SMN2L3MBTL1RECQLADORA3ADORA2A
SCHEMBL30412355 0.76 KDR (0.70) NPSR1CA1CA2CA9
SCHEMBL19668006 0.76 KDR (0.70) NPSR1CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5877191-A ANTIINFLAMMATORY AGENT; ANALGESICS; ANTIHISTAMINES; EMESIS MERCK & CO., INC. (US) 1999-03-02 US disclosed
WO-1998017660-A1 PHENYL SPIROETHERCYCLOALKYL TACHYKININ RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1998-04-30 WO disclosed