SCHEMBL8519455

SCHEMBL8519455

Cc1ccccc1C(=O)CN1CC(=O)N=Cc2ccccc21

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTNNB1 P35222 4/20 0.39
WNT3A P56704 4/20 0.39
ERCC5 P28715 1/20 0.38
FEN1 P39748 1/20 0.38
BCHE P06276 1/20 0.35
HTT P42858 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
KMT2A Q03164 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34
TSHR P16473 1/20 0.33
ATM Q13315 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7480896 0.78 ALDH1A1 (0.41) HTTL3MBTL1MEN1NPC1RAB9A
SCHEMBL7484284 0.77 HSD17B3 (0.35) L3MBTL1MEN1KMT2ATSHR
SCHEMBL6584861 0.67 ERCC5 (0.39) CTNNB1WNT3AERCC5FEN1BCHE
SCHEMBL11813934 0.66 KMT2A (0.62) HTTL3MBTL1MEN1NPC1RAB9A
SCHEMBL8735550 0.62 ERCC5 (0.74) CTNNB1WNT3AERCC5FEN1L3MBTL1
SCHEMBL30089517 0.62 CTNNB1 (0.68) CTNNB1WNT3AERCC5FEN1L3MBTL1
SCHEMBL15979740 0.62 CTNNB1 (0.68) CTNNB1WNT3AERCC5FEN1L3MBTL1
SCHEMBL13161999 0.61 ALDH1A1 (0.60) HTTL3MBTL1MEN1RAB9AKMT2A
SCHEMBL31901342 0.61 ERCC5 (0.60) CTNNB1WNT3AERCC5FEN1L3MBTL1
SCHEMBL3704844 0.61 ERCC5 (0.60) CTNNB1WNT3AERCC5FEN1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934282-A1 1,4-BENZODIAZEPINONES AND THEIR USES AS CCK ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-08-11 EP disclosed
WO-1998015535-A1 1,4-BENZODIAZEPINONES AND THEIR USES AS CCK ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-04-16 WO disclosed