SCHEMBL8520030

SCHEMBL8520030

CC(C(=O)O)N1CCCN(c2ccccc2)C1=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
KMT2A Q03164 2/20 0.49
CYP2D6 P10635 3/20 0.40
CYP1A2 P05177 2/20 0.40
CYP2C9 P11712 2/20 0.40
KDM4E B2RXH2 1/20 0.38
DRD2 P14416 1/20 0.38
DRD3 P35462 1/20 0.38
DDB1 Q16531 1/20 0.38
CRBN Q96SW2 1/20 0.38
PER2 O15055 2/20 0.38
CRY2 Q49AN0 1/20 0.38
TP53 P04637 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
CYP2C19 P33261 2/20 0.37
CYP3A4 P08684 2/20 0.37
ACE P12821 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8411315 0.91 MEN1 (0.56) MEN1NPC1RAB9AKMT2ACYP2D6
SCHEMBL6362002 0.76 NPC1 (0.82) MEN1NPC1RAB9AKMT2AKDM4E
SCHEMBL11036674 0.74 MEN1 (0.55) MEN1NPC1RAB9AKMT2AKDM4E
SCHEMBL8026728 0.74 MEN1 (0.64) MEN1NPC1RAB9AKMT2ADRD2
SCHEMBL6362778 0.72 MEN1 (0.61) MEN1NPC1RAB9AKMT2AKDM4E
SCHEMBL8397598 0.71 MEN1 (0.50) MEN1NPC1RAB9AKMT2ACYP2D6
SCHEMBL4515174 0.70 KMT2A (0.58) MEN1NPC1RAB9AKMT2ACYP2D6
SCHEMBL8520034 0.69 RAB9A (0.40) MEN1NPC1RAB9AKMT2ACYP2D6
SCHEMBL14019897 0.69 MEN1 (0.51) MEN1NPC1RAB9AKMT2ACYP2D6
SCHEMBL909200 0.68 MEN1 (0.61) MEN1NPC1RAB9AKMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0932598-A1 ASPARTATE ESTER INHIBITORS OF INTERLEUKIN-1$g(b) CONVERTING ENZYME WARNER-LAMBERT COMPANY (US) 1999-08-04 EP disclosed
WO-1998016502-A1 ASPARTATE ESTER INHIBITORS OF INTERLEUKIN-1β CONVERTING ENZYME WARNER-LAMBERT COMPANY (US) 1998-04-23 WO disclosed