SCHEMBL8520674

SCHEMBL8520674

Cc1cc(C(=O)NC2CC(=O)c3ccccc3N(CC(=O)OCc3ccccc3)C2=O)cc(C)c1O

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 4/20 0.42
CCKAR P32238 3/20 0.39
PYGL P06737 1/20 0.38
SENP1 Q9P0U3 1/20 0.37
HTR1A P08908 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5712951 1.00 CCKBR (0.42) CCKBRCCKARPYGLSENP1HTR1A
SCHEMBL5712995 0.87 PYGL (0.44) CCKBRCCKARPYGLHTR1A
SCHEMBL5712987 0.81 CCKBR (0.45) CCKBR
SCHEMBL8521032 0.81 CCKBR (0.45) CCKBR
SCHEMBL7446421 0.78 CASP1 (0.39) CCKBRPYGL
SCHEMBL6674788 0.77 CASP1 (0.46) CCKBR
SCHEMBL8520881 0.77 CASP1 (0.46) CCKBR
Hydrochloric Acid SCHEMBL5713016 0.74 CCKBR (0.46) CCKBRCCKARSENP1
SCHEMBL646039 0.73 CASP1 (0.50) CCKBR
SCHEMBL7568437 0.72 CCKBR (0.46) CCKBRCCKAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0942925-A2 INHIBITORS OF INTERLEUKIN-1$g(b) CONVERTING ENZYME Vertex Pharmaceuticals Incorporated (US) 1999-09-22 EP disclosed
WO-1998024804-A2 INHIBITORS OF INTERLEUKIN-1β CONVERTING ENZYME VERTEX PHARMACEUTICALS INCORPORATED (US) 1998-06-11 WO disclosed