SCHEMBL852142

SCHEMBL852142

NS(=O)(=O)c1ccc2oc(=O)c(S(N)(=O)=O)cc2c1

nearest known ligand 0.69

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CA12 O43570 12/20 0.69
CA1 P00915 12/20 0.69
CA9 Q16790 12/20 0.69
CA2 P00918 11/20 0.69
PKM P14618 4/20 0.51
ALPL P05186 1/20 0.51
ALPI P09923 1/20 0.51
RXFP1 Q9HBX9 1/20 0.50
LMNA P02545 3/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27792013 0.82 CA12 (1.00) CA12CA1CA9CA2PKM
SCHEMBL8810276 0.80 CA12 (1.00) CA12CA1CA9CA2LMNA
SCHEMBL830136 0.79 CA1 (1.00) CA12CA1CA9CA2RXFP1
SCHEMBL31287831 0.76 SMN1; SMN2 (0.56) CA12CA1CA9CA2PKM
SCHEMBL1743537 0.76 SMN1; SMN2 (0.56) CA12CA1CA9CA2PKM
Furan SCHEMBL1680246 0.73 CA1 (0.85) CA12CA1CA9CA2RXFP1
SCHEMBL830157 0.71 CA2 (0.56) CA12CA1CA9CA2PKM
SCHEMBL21033100 0.70 CA12 (0.68) CA12CA1CA9CA2PKM
SCHEMBL20435633 0.70 LMNA (0.80) CA12CA1CA9CA2PKM
SCHEMBL5428747 0.69 GPR27 (0.56) CA12CA1CA9CA2PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143428-B2 Heteroaryl sulfones and sulfonamides and therapeutic uses thereof TEMPLE UNIVERSITY-OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2012-03-27 US disclosed
US-20070232649-A1 Heteroaryl Sulfones and Sulfonamides and Therapeutic Uses Thereof TEMPLE UNIVERSITY-OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2007-10-04 US disclosed
EP-1765804-A2 HETEROARYL SULFONES AND SULFONAMIDES AND THERAPEUTIC USES THEREOF Temple University of the Commonwealth System of Higher Education (US) 2007-03-28 EP disclosed
WO-2005123077-A2 HETEROARYL SULFONES AND SULFONAMIDES AND THERAPEUTIC USES THEREOF TEMPLE UNIVERSITY-OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2005-12-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070232649-A1 Heteroaryl Sulfones and Sulfonamides and Therapeutic Uses Thereof SULT1E1, STS, CCNE1 CA12 2448/4885CA1 3859/4885CA9 1884/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.