SCHEMBL8521983

SCHEMBL8521983

C#Cc1scc(C(=O)ON)c1N(Cc1ccccc1)S(=O)(=O)c1ccc(OC)cc1

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MMP9 P14780 16/20 0.58
MMP13 P45452 15/20 0.58
MMP1 P03956 13/20 0.58
ADAM17 P78536 3/20 0.52
LMNA P02545 2/20 0.48
NR3C1 P04150 1/20 0.48
PGR P06401 1/20 0.48
ALDH1A1 P00352 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
MAPT P10636 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6559690 0.93 MMP9 (0.63) MMP9MMP13MMP1ADAM17LMNA
Hydroxyamine SCHEMBL8521982 0.91 MMP9 (0.60) MMP9MMP13MMP1ADAM17LMNA
SCHEMBL6558860 0.91 MMP9 (0.62) MMP9MMP13MMP1ADAM17LMNA
SCHEMBL7467779 0.87 MMP9 (0.78) MMP9MMP13MMP1ADAM17
SCHEMBL7463546 0.80 MMP9 (0.59) MMP9MMP13MMP1ADAM17
SCHEMBL6561291 0.79 MMP9 (0.83) MMP9MMP13MMP1ADAM17
SCHEMBL8521996 0.79 MMP9 (0.56) MMP9MMP13MMP1ADAM17LMNA
SCHEMBL7413282 0.78 MMP9 (0.52) MMP9MMP13MMP1ADAM17LMNA
SCHEMBL6560148 0.76 MMP9 (0.83) MMP9MMP13MMP1ADAM17LMNA
SCHEMBL7315545 0.75 MMP13 (0.65) MMP9MMP13MMP1ADAM17

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934300-A1 THE PREPARATION AND USE OF ORTHO-SULFONAMIDO HETEROARYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE AND TACE INHIBITORS American Cyanamid Company (US) 1999-08-11 EP disclosed
WO-1998016520-A1 THE PREPARATION AND USE OF ORTHO-SULFONAMIDO HETEROARYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE AND TACE INHIBITORS AMERICAN CYANAMID COMPANY (US) 1998-04-23 WO disclosed