SCHEMBL8523260

SCHEMBL8523260

Cc1nnc2n1-c1ccccc1N(CCCN1CCC(C(O)(c3cccs3)c3cccs3)CC1)C2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 5/20 0.37
KCNH2 Q12809 4/20 0.37
CYP2J2 P51589 3/20 0.35
KDM1A O60341 1/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
AVPR2 P30518 2/20 0.33
NPC1 O15118 1/20 0.33
CACNA1F O60840 1/20 0.33
GMNN O75496 1/20 0.33
USP2 O75604 1/20 0.33
EGFR P00533 1/20 0.33
LMNA P02545 1/20 0.33
CYP1A2 P05177 1/20 0.33
FYN P06241 1/20 0.33
CHRM2 P08172 1/20 0.33
ABCB1 P08183 1/20 0.33
CYP3A4 P08684 1/20 0.33
HTR1A P08908 1/20 0.33
ADRA2A P08913 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8317297 0.84 HRH1 (0.39) HRH1KCNH2CYP2J2MEN1KMT2A
SCHEMBL8317429 0.82 HRH1 (0.39) HRH1KCNH2CYP2J2MEN1KMT2A
SCHEMBL8316037 0.82 HRH1 (0.46) HRH1KCNH2CYP2J2MEN1KMT2A
SCHEMBL8315418 0.81 PAX8 (0.40) HRH1KCNH2CYP2J2AVPR2HTR1A
SCHEMBL8312317 0.81 HRH1 (0.48) HRH1KCNH2CYP2J2MEN1KMT2A
SCHEMBL8315211 0.81 HRH1 (0.46) HRH1KCNH2CYP2J2MEN1KMT2A
SCHEMBL8317157 0.79 CYP2J2 (0.45) HRH1KCNH2CYP2J2MEN1KMT2A
SCHEMBL8315487 0.79 CYP2J2 (0.39) HRH1KCNH2CYP2J2MEN1KMT2A
SCHEMBL8314774 0.78 CYP2J2 (0.47) HRH1KCNH2CYP2J2MEN1KMT2A
SCHEMBL8313333 0.77 HRH1 (0.43) HRH1KCNH2CYP2J2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0536419-B1 TRICYCLIC TRIAZOLE DERIVATIVES, PRODUCTION AND USE THEREOF TORAY INDUSTRIES (JP) 1999-10-13 EP disclosed
EP-0536419-A1 TRICYCLIC TRIAZOLE DERIVATIVE, PRODUCTION THEREOF, AND USE THEREOF TORAY INDUSTRIES, INC. (JP) 1993-04-14 EP disclosed