SCHEMBL8524150

SCHEMBL8524150

CS(=O)(=O)Nc1cc(CO)c(N)cc1Oc1ccc(Cl)cc1Cl

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 2/20 0.54
PTGS2 P35354 2/20 0.54
CCR2 P41597 1/20 0.47
CYP2C9 P11712 1/20 0.44
SLC6A3 Q01959 8/20 0.42
SLC6A4 P31645 8/20 0.42
SLC6A2 P23975 8/20 0.42
KCNH2 Q12809 3/20 0.42
HPGD P15428 2/20 0.42
ALDH1A1 P00352 1/20 0.42
POLB P06746 1/20 0.42
GAA P10253 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
TTR P02766 2/20 0.41
CHRM1 P11229 1/20 0.39
NR1I2 O75469 1/20 0.39
LMNA P02545 1/20 0.39
PGR P06401 1/20 0.39
HSP90AA1 P07900 1/20 0.39
ADORA3 P0DMS8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8101582 0.89 PTGS1 (0.50) PTGS1PTGS2CCR2CYP2C9SLC6A3
SCHEMBL8525177 0.83 PTGS1 (0.50) PTGS1PTGS2CCR2CYP2C9SLC6A3
SCHEMBL8523577 0.81 PTGS1 (0.58) PTGS1PTGS2CCR2CYP2C9SLC6A3
SCHEMBL8524769 0.79 PTGS1 (0.50) PTGS1PTGS2CCR2CYP2C9SLC6A3
SCHEMBL8099718 0.74 PTGS1 (0.68) PTGS1PTGS2CCR2SLC6A3SLC6A4
SCHEMBL8107162 0.74 PTGS1 (0.61) PTGS1PTGS2CCR2CYP2C9SLC6A3
SCHEMBL9657545 0.74 PTGS1 (0.61) PTGS1PTGS2CCR2SLC6A3SLC6A4
SCHEMBL11177507 0.74 PTGS2 (0.58) PTGS1PTGS2CCR2CYP2C9SLC6A3
SCHEMBL8101589 0.74 PTGS2 (0.61) PTGS1PTGS2CCR2CYP2C9SLC6A3
Methylamine SCHEMBL8479365 0.74 PTGS2 (0.58) PTGS1PTGS2CCR2CYP2C9SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6004948-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS; SIDE EFFECT REDUCTION NYCOMED AUSTRIA GMBH (AT) 1999-12-21 US disclosed