SCHEMBL8524248

SCHEMBL8524248

OC1C(I)C[C@H](n2cnc3cc(Cl)c(Cl)cc32)C1O

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.41
AHCY P23526 9/20 0.36
CYP2C9 P11712 1/20 0.36
IDO1 P14902 1/20 0.36
KCNH2 Q12809 1/20 0.36
PRPS1 P60891 2/20 0.36
IRAK4 Q9NWZ3 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8524247 1.00 THRB (0.41) THRBAHCYCYP2C9IDO1KCNH2
SCHEMBL9119445 0.81 AHCY (0.57) THRBAHCY
SCHEMBL8525972 0.81 AHCY (0.57) THRBAHCY
SCHEMBL8525973 0.81 AHCY (0.57) THRBAHCY
SCHEMBL9120372 0.81 AHCY (0.57) THRBAHCY
SCHEMBL9120465 0.81 AHCY (0.57) THRBAHCY
SCHEMBL8659894 0.77 AHCY (0.52) THRBAHCYCYP2C9IDO1KCNH2
SCHEMBL8659891 0.77 AHCY (0.52) THRBAHCYCYP2C9IDO1KCNH2
SCHEMBL7616161 0.75 PRPS1 (0.48) THRBKCNH2PRPS1
SCHEMBL7616155 0.75 PRPS1 (0.48) THRBKCNH2PRPS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5912356-A HERPES VIRUS GLAXO WELLCOME INC. (US) 1999-06-15 US disclosed
EP-0779885-A1 ANTIVIRAL NUCLEOSIDE ANALOGUES CONTAINING A SUBSTITUTED BENZIMIDAZOLE BASE ATTACHED TO A CARBOCYCLIC RING THE WELLCOME FOUNDATION LIMITED (GB) 1997-06-25 EP disclosed
US-5534535-A ANTIVIRAL ANALOGS WITH SUBSTITUTED BENZIMIDAZOLE BASE BURROUGHS WELLCOME CO. (US) 1996-07-09 US disclosed
WO-1996007646-A1 ANTIVIRAL NUCLEOSIDE ANALOGUES CONTAINING A SUBSTITUTED BENZIMIDAZOLE BASE ATTACHED TO A CARBOCYCLIC RING THE WELLCOME FOUNDATION LIMITED (GB) 1996-03-14 WO disclosed