SCHEMBL8525580

SCHEMBL8525580

COc1ccc(/C(=C/C#N)c2cccc3ccccc23)cc1OC.COc1ccc(C(=O)c2cccc3ccccc23)cc1OC

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 16/20 0.57
PDE4B Q07343 16/20 0.57
PDE4C Q08493 16/20 0.57
PDE4D Q08499 16/20 0.57
AKR1C2 P52895 1/20 0.48
ALDH1A1 P00352 1/20 0.48
GAA P10253 1/20 0.48
MAPT P10636 1/20 0.48
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
TSHR P16473 1/20 0.45
CYP2C19 P33261 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8525581 1.00 PDE4A (0.57) PDE4APDE4BPDE4CPDE4DAKR1C2
SCHEMBL4818722 0.93 PDE4A (0.66) PDE4APDE4BPDE4CPDE4DAKR1C2
SCHEMBL4818718 0.93 PDE4A (0.66) PDE4APDE4BPDE4CPDE4DAKR1C2
SCHEMBL5077492 0.86 ALDH1A1 (0.61) AKR1C2ALDH1A1GAAMAPTCYP1A2
SCHEMBL10848469 0.78 PDE4A (0.44) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL10848465 0.78 PDE4A (0.44) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL28816702 0.78 PDE4A (0.71) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL13984813 0.77 PDE4A (0.69) PDE4APDE4BPDE4CPDE4D
SCHEMBL13986023 0.77 PDE4A (0.69) PDE4APDE4BPDE4CPDE4D
SCHEMBL4824892 0.76 PDE4A (0.78) PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0918746-A1 IMMUNOTHERAPEUTIC AGENTS AND THEIR USE IN THE REDUCTION OF CYTOKINE LEVELS CELGENE CORPORATION (US) 1999-06-02 EP disclosed
WO-1998006692-A1 NOVEL IMMUNOTHERAPEUTIC AGENTS AND THEIR USE IN THE REDUCTION OF CYTOKINE LEVELS CELGENE CORPORATION (US) 1998-02-19 WO disclosed