SCHEMBL8525879

SCHEMBL8525879

O=C(O)CCC1=CC(F)=CC(F)(c2cccc(NS(=O)(=O)c3cccc(NC4=NCCN4)c3)c2)C1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 9/20 0.41
ITGAV P06756 9/20 0.41
ITGA2B P08514 8/20 0.41
ITGB1 P05556 3/20 0.37
ITGB5 P18084 3/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.33
ALDH1A1 P00352 2/20 0.32
ADRA2A P08913 1/20 0.32
ADRA2B P18089 1/20 0.32
ADRA2C P18825 1/20 0.32
AURKA O14965 1/20 0.32
AURKB Q96GD4 1/20 0.32
MITF O75030 1/20 0.31
POLB P06746 1/20 0.31
PTGIR P43119 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8500892 0.81 PTGDR2 (0.35) PTGDR2ALDH1A1POLB
SCHEMBL8526327 0.77 ITGB3 (0.49) ITGB3ITGAVITGA2BITGB1ITGB5
SCHEMBL6798729 0.71 ITGB3 (0.44) ITGB3ITGAVITGA2BITGB1ITGB5
SCHEMBL7785708 0.68 ITGB3 (0.53) ITGB3ITGAVITGA2BITGB1ITGB5
SCHEMBL8501256 0.67 KMT2A (0.33) PTGDR2POLB
SCHEMBL7997106 0.66 ITGB3 (0.70) ITGB3ITGAVITGA2BITGB1ITGB5
SCHEMBL7856513 0.66 ITGB3 (0.45) ITGB3ITGAVITGA2BITGB1ITGB5
SCHEMBL8532462 0.65 ITGB3 (0.43) ITGB3ITGAVITGA2BITGB1ITGB5
SCHEMBL7367300 0.64 ITGB3 (0.51) ITGB3ITGAVITGA2BITGB1ITGB5
SCHEMBL8532458 0.63 ITGB3 (0.40) ITGB3ITGAVITGA2BITGB1ITGB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1999-01-13 EP claimed
WO-1997036862-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1997-10-09 WO claimed