SCHEMBL8526592

SCHEMBL8526592

CC(c1ccccc1OCc1ccccc1)N(CC=O)C(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
ALDH1A1 P00352 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
RXRA P19793 1/20 0.39
RXRB P28702 1/20 0.39
RXRG P48443 1/20 0.39
BRD4 O60885 1/20 0.38
ITGA4 P13612 1/20 0.38
ITGB7 P26010 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
PTGER1 P34995 3/20 0.38
PTGER4 P35408 3/20 0.38
PTGER3 P43115 3/20 0.38
PTGER2 P43116 3/20 0.38
MME P08473 1/20 0.37
ACE P12821 1/20 0.37
CPA1 P15085 1/20 0.37
ACE2 Q9BYF1 1/20 0.37
CCNB2 O95067 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8542129 0.76 PTGER1 (0.47) L3MBTL1PTGER1PTGER4PTGER3PTGER2
SCHEMBL7413567 0.74 POLB (0.43) ALDH1A1L3MBTL1NPSR1
SCHEMBL7413529 0.74 POLB (0.43) ALDH1A1L3MBTL1NPSR1
SCHEMBL8502030 0.74 NPSR1 (0.47) L3MBTL1NPSR1
SCHEMBL7351228 0.73 ATM (0.42) L3MBTL1ITGA4ITGB7NPSR1ACE
SCHEMBL8770890 0.72 RXRA (0.43) KDM4ETDP1L3MBTL1RXRARXRB
SCHEMBL27984256 0.71 SYK (0.51) ALDH1A1BRD4ACE
SCHEMBL1845821 0.71 HTR1A (0.48) KDM4ETDP1ALDH1A1L3MBTL1RXRA
SCHEMBL8132061 0.70 MRGPRX4 (0.40) ALDH1A1L3MBTL1
SCHEMBL29575338 0.70 PPARA (0.53) ACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5864045-A Heterocyclic substituted piperazinone derivatives HOECHST MARION ROUSSEL, INC. (US) 1999-01-26 US disclosed
US-5840726-A Heterocyclic substituted piperazinone derivatives HOECHST MARION ROUSSEL INC. (US) 1998-11-24 US disclosed