SCHEMBL8542129

SCHEMBL8542129

CC(C)(C)OC(=O)N(CC=O)CCc1ccccc1OCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 2/20 0.47
PTGER4 P35408 2/20 0.47
PTGER3 P43115 2/20 0.47
PTGER2 P43116 2/20 0.47
HTR1A P08908 2/20 0.46
DRD2 P14416 2/20 0.46
BCHE P06276 4/20 0.43
ABCB1 P08183 3/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
SLC1A5 Q15758 2/20 0.41
GAA P10253 1/20 0.41
FOLH1 Q04609 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8540237 0.90 BCHE (0.52) PTGER1PTGER4PTGER3PTGER2HTR1A
SCHEMBL1846485 0.84 MEN1 (0.44) L3MBTL1
SCHEMBL7835952 0.84 LTB4R (0.52) BCHEL3MBTL1
SCHEMBL7646792 0.82 HTR1A (0.51) PTGER1PTGER4PTGER3PTGER2HTR1A
SCHEMBL4289433 0.81 L3MBTL1 (0.44) HTR1AL3MBTL1
SCHEMBL2722481 0.77 HDAC3 (0.53) L3MBTL1
SCHEMBL1845821 0.76 HTR1A (0.48) PTGER1PTGER4PTGER3PTGER2HTR1A
SCHEMBL8526592 0.76 KDM4E (0.40) PTGER1PTGER4PTGER3PTGER2L3MBTL1
SCHEMBL31153832 0.75 L3MBTL1 (0.43) L3MBTL1
SCHEMBL22513467 0.75 MEN1 (0.51) PTGER1PTGER4PTGER3PTGER2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0815105-A1 HETEROCYCLIC SUBSTITUTED PIPERAZINONE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS HOECHST MARION ROUSSEL, INC. (US) 1998-01-07 EP disclosed
WO-1996028441-A1 HETEROCYCLIC SUBSTITUTED PIPERAZINONE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS HOECHST MARION ROUSSEL, INC. (US) 1996-09-19 WO disclosed