SCHEMBL8527555

SCHEMBL8527555

CC(C)(C)OC(=O)N[C@@H](Cc1ccc([N+](=O)[O-])s1)C(=O)OC(C)(C)C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
ALDH1A1 P00352 2/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
NR1D1 P20393 9/20 0.45
NR1H3 Q13133 1/20 0.44
GSTP1 P09211 1/20 0.43
GSTM2 P28161 1/20 0.43
CTSS P25774 3/20 0.42
CTSK P43235 2/20 0.42
PPARG P37231 1/20 0.41
PPARA Q07869 1/20 0.41
ITGA4 P13612 1/20 0.41
ITGB7 P26010 1/20 0.41
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HTT P42858 2/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8527559 1.00 MAPT (0.48) MAPTSMN1; SMN2ALDH1A1MEN1KMT2A
SCHEMBL8423298 0.92 MAPT (0.46) MAPTSMN1; SMN2ALDH1A1MEN1KMT2A
SCHEMBL8423297 0.92 MAPT (0.46) MAPTSMN1; SMN2ALDH1A1MEN1KMT2A
SCHEMBL8528928 0.81 NR1D1 (0.48) MAPTSMN1; SMN2ALDH1A1MEN1KMT2A
SCHEMBL8528925 0.81 NR1D1 (0.48) MAPTSMN1; SMN2ALDH1A1MEN1KMT2A
SCHEMBL8530056 0.81 CTSS (0.45) MAPTALDH1A1CTSSCTSKKDM4E
SCHEMBL8530060 0.81 CTSS (0.45) MAPTALDH1A1CTSSCTSKKDM4E
SCHEMBL8422157 0.81 CTSS (0.45) CTSSCTSKCTSLCTSB
SCHEMBL8422158 0.81 CTSS (0.45) CTSSCTSKCTSLCTSB
SCHEMBL3784750 0.77 PPARG (0.59) MAPTSMN1; SMN2ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705257-B1 AMINOACID DERIVATIVES AS NO SYNTHASE INHIBITORS WELLCOME FOUND (GB) 1998-03-11 EP disclosed