SCHEMBL8528161

SCHEMBL8528161

CCC(CC)C(=O)NC(Cc1ccccc1)(C(=O)O)C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.48
RECQL P46063 2/20 0.48
KMT2A Q03164 2/20 0.45
MEN1 O00255 1/20 0.45
PKM P14618 1/20 0.44
CYP3A4 P08684 2/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
TSHR P16473 1/20 0.43
ENPEP Q07075 2/20 0.43
HIF1A Q16665 1/20 0.42
MMP8 P22894 1/20 0.42
CYP1A2 P05177 2/20 0.41
ADORA1 P30542 1/20 0.40
LMNA P02545 1/20 0.40
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8421523 0.86 KMT2A (0.39) ALDH1A1RECQLKMT2AMEN1PKM
SCHEMBL9503704 0.85 KMT2A (0.64) ALDH1A1RECQLKMT2APKMCYP3A4
SCHEMBL8526626 0.82 ALDH1A1 (0.49) ALDH1A1KMT2AMEN1CYP2C19SMN1; SMN2
SCHEMBL8954953 0.82 FOLH1 (0.43) KMT2APKMADORA1LMNA
SCHEMBL8426514 0.81 ALDH1A1 (0.46) ALDH1A1RECQLKMT2AMEN1CYP2C9
SCHEMBL8423454 0.80 LMNA (0.40) ALDH1A1KMT2AMEN1PKMSMN1; SMN2
SCHEMBL8422033 0.79 LMNA (0.44) KMT2AMEN1PKMTSHRLMNA
SCHEMBL28168069 0.78 ALDH1A1 (0.67) ALDH1A1RECQLCYP3A4CYP2C9CYP2C19
SCHEMBL1196133 0.76 TSHR (0.45) ALDH1A1KMT2AMEN1PKMSMN1; SMN2
SCHEMBL6512076 0.74 KMT2A (0.44) ALDH1A1KMT2AMEN1CYP3A4SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705257-B1 AMINOACID DERIVATIVES AS NO SYNTHASE INHIBITORS WELLCOME FOUND (GB) 1998-03-11 EP disclosed
EP-0705257-A1 AMINOACID DERIVATIVES AS NO SYNTHASE INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1996-04-10 EP disclosed
WO-1995000505-A1 AMINOACID DERIVATIVES AS NO SYNTHASE INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1995-01-05 WO disclosed