SCHEMBL8528753

SCHEMBL8528753

CSc1cc2c(cc1Br)NCC2

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.45
MAPT P10636 1/20 0.45
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
HTR2A P28223 3/20 0.33
HTR2C P28335 3/20 0.33
AR P10275 2/20 0.33
GFER P55789 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HTR2B P41595 1/20 0.32
PARP10 Q53GL7 2/20 0.31
PARP11 Q9NR21 1/20 0.31
PARP1 P09874 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8785768 0.85 ALDH1A1 (0.47) ALDH1A1MAPTDRD2DRD4HTR2A
SCHEMBL8527738 0.81 ALDH1A1 (0.42) ALDH1A1MAPTDRD2DRD4AR
SCHEMBL8526682 0.79 ALDH1A1 (0.40) ALDH1A1MAPTDRD2DRD4SMN1; SMN2
SCHEMBL3238397 0.79 DRD2 (0.42) ALDH1A1MAPTDRD2DRD4HTR2A
SCHEMBL6187333 0.79 DRD2 (0.38) ALDH1A1MAPTDRD2DRD4HTR2A
SCHEMBL3237859 0.79 DRD2 (0.38) ALDH1A1MAPTDRD2DRD4HTR2A
SCHEMBL3242042 0.76 HTR2A (0.40) ALDH1A1MAPTDRD2DRD4HTR2A
SCHEMBL3731583 0.76 ALDH1A1 (0.49) ALDH1A1MAPTDRD2DRD4HTR2A
SCHEMBL7079658 0.75 AR (0.48) ALDH1A1MAPTDRD2DRD4HTR2A
Hydrochloric Acid SCHEMBL7078884 0.73 DRD2 (0.34) ALDH1A1MAPTDRD2DRD4AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5834494-A SEROTONIN 5HT2B/2C RECEPTOR ANTAGONISTS; CNS NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS; IRRITABLE BOWEL SYNDROME SMITHKLINE BEECHAM P.L.C. (GB) 1998-11-10 US disclosed
EP-0707581-B1 INDOLINE DERIVATIVES AS 5HT2C ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1997-02-26 EP disclosed
EP-0707581-A1 INDOLINE DERIVATIVES AS 5HT 2C? ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1996-04-24 EP disclosed
WO-1995001976-A1 INDOLINE DERIVATIVES AS 5HT2C ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1995-01-19 WO disclosed