SCHEMBL8528962

SCHEMBL8528962

COC(=O)Cc1c[nH]c2ccc(C(=O)OC)cc12

nearest known ligand 0.68

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 1/20 0.68
NPC1 O15118 1/20 0.56
KDM4E B2RXH2 2/20 0.52
HTR7 P34969 2/20 0.49
HTR6 P50406 1/20 0.49
KMT2A Q03164 2/20 0.49
MEN1 O00255 1/20 0.49
ATM Q13315 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
HTR1A P08908 1/20 0.49
HTR1D P28221 1/20 0.49
HTR1B P28222 1/20 0.49
CDK2 P24941 1/20 0.47
POLB P06746 1/20 0.47
MTNR1A P48039 1/20 0.47
MTNR1B P49286 1/20 0.47
ALDH1A1 P00352 1/20 0.47
HPGD P15428 1/20 0.47
HSD17B10 Q99714 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31571584 0.89 GPR84 (0.68) GPR84NPC1KDM4EHTR7HTR6
SCHEMBL27142546 0.89 GPR84 (0.68) GPR84NPC1KDM4EHTR7HTR6
SCHEMBL29871648 0.87 GPR84 (0.87) GPR84NPC1KDM4EHTR7HTR6
SCHEMBL22554662 0.87 GPR84 (0.73) GPR84NPC1KDM4EHTR7HTR6
SCHEMBL2161423 0.86 GPR84 (0.76) GPR84NPC1KDM4EHTR7HTR6
SCHEMBL2161735 0.84 GPR84 (0.70) GPR84NPC1KDM4EHTR7HTR6
SCHEMBL3974212 0.83 NPC1 (0.80) GPR84NPC1KDM4EHTR7HTR6
SCHEMBL10174674 0.83 HTR1D (0.56) GPR84KDM4EHTR1AHTR1DHTR1B
SCHEMBL12844152 0.83 GPR84 (0.68) GPR84NPC1HTR7HTR6KMT2A
SCHEMBL853729 0.83 NPSR1 (0.68) KDM4EHTR7HTR6KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0489547-B1 A process for the preparation of a 3-alkylated indole, intermediates, and a process for the preparation of a derivative thereof ZENECA LTD (GB) 1998-07-29 EP disclosed
US-5280125-A Chemical process for the preparation of 3-alkylated indole IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1994-01-18 US disclosed
EP-0489547-A1 A process for the preparation of a 3-alkylated indole, intermediates, and a process for the preparation of a derivative thereof ZENECA LIMITED (GB) 1992-06-10 EP disclosed