SCHEMBL8529274

SCHEMBL8529274

COc1nc(N)nc2c1ncn2[C@@H]1O[C@H](CO)[C@@H](OC(C)=O)[C@@H]1OC(C)=O

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.53
LMNA P02545 1/20 0.53
TP53 P04637 1/20 0.53
MAPT P10636 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
CYP2C19 P33261 1/20 0.48
ADORA2A P29274 3/20 0.48
ADORA3 P0DMS8 2/20 0.48
ADORA1 P30542 2/20 0.48
ADORA2B P29275 2/20 0.48
SLC29A1 Q99808 6/20 0.46
PGK1 P00558 1/20 0.44
PGK2 P07205 1/20 0.44
ACHE P22303 2/20 0.43
HINT1 P49773 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8530540 0.92 CYP2C19 (0.54) ALDH1A1LMNATP53MAPTTDP1
SCHEMBL8527967 0.90 ALDH1A1 (0.66) ALDH1A1LMNATP53MAPTTDP1
SCHEMBL13743273 0.89 ALDH1A1 (0.56) ALDH1A1LMNATP53MAPTTDP1
SCHEMBL8529155 0.86 ALDH1A1 (0.52) ALDH1A1LMNATP53MAPTTDP1
SCHEMBL8532634 0.85 ALDH1A1 (0.57) ALDH1A1LMNATP53MAPTTDP1
SCHEMBL8531895 0.83 ALDH1A1 (0.57) ALDH1A1LMNATP53MAPTTDP1
SCHEMBL8529436 0.82 ALDH1A1 (0.48) ALDH1A1LMNATP53MAPTTDP1
SCHEMBL8532515 0.82 CYP2C19 (0.52) CYP2C19ADORA2AADORA3ADORA1ADORA2B
SCHEMBL8529892 0.82 CYP2C19 (0.52) CYP2C19ADORA2AADORA3ADORA1ADORA2B
SCHEMBL17198372 0.82 ALDH1A1 (0.47) ALDH1A1LMNATP53MAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5821236-A Tumor treatment with arabinofuranosyl purine derivatives GLAXO WELLCOME INC. (US) 1998-10-13 US claimed
EP-0539479-B1 HETEROCYCLIC COMPOUNDS WELLCOME FOUND (GB) 1997-04-16 EP claimed
US-5821236-A Tumor treatment with arabinofuranosyl purine derivatives GLAXO WELLCOME INC. (US) 1998-10-13 US disclosed
US-5747472-A ANTICARCINOGENIC AGENTS AND ANTITUMOR AGENTS GLAXO WELLCOME INC. (US) 1998-05-05 US disclosed
EP-0539479-B1 HETEROCYCLIC COMPOUNDS WELLCOME FOUND (GB) 1997-04-16 EP disclosed
US-5492897-A ANTITUMOR AGENTS, AUTOIMMUNE DISEASES BURROUGHS WELLCOME CO. (141) (US) 1996-02-20 US disclosed
WO-1992001456-A1 HETEROCYCLIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1992-02-06 WO disclosed