SCHEMBL8529155

SCHEMBL8529155

COc1nc(N)nc2c1ncn2[C@@H]1O[C@H](CO[Si](C)(C)C(C)(C)C)[C@@H](OC(C)=O)[C@@H]1OC(C)=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
LMNA P02545 1/20 0.52
TP53 P04637 1/20 0.52
MAPT P10636 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
HINT1 P49773 2/20 0.42
PRKAB2 O43741 1/20 0.41
PRKAG1 P54619 1/20 0.41
PRKAA2 P54646 1/20 0.41
PRKAA1 Q13131 1/20 0.41
PRKAG3 Q9UGI9 1/20 0.41
PRKAG2 Q9UGJ0 1/20 0.41
PRKAB1 Q9Y478 1/20 0.41
ACHE P22303 3/20 0.40
NT5E P21589 2/20 0.40
CYP2C19 P33261 1/20 0.38
HSP90B1 P14625 1/20 0.38
ADORA3 P0DMS8 3/20 0.37
ADORA1 P30542 2/20 0.37
ADORA2B P29275 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8529436 0.96 ALDH1A1 (0.48) ALDH1A1LMNATP53MAPTTDP1
SCHEMBL8533171 0.88 HINT1 (0.40) ALDH1A1LMNATP53MAPTTDP1
SCHEMBL8529887 0.88 HINT1 (0.40) ALDH1A1LMNATP53MAPTTDP1
SCHEMBL8527967 0.88 ALDH1A1 (0.66) ALDH1A1LMNATP53MAPTTDP1
SCHEMBL8533343 0.87 HINT1 (0.40) ALDH1A1LMNATP53MAPTTDP1
SCHEMBL8529274 0.86 ALDH1A1 (0.53) ALDH1A1LMNATP53MAPTTDP1
SCHEMBL8988189 0.86 HINT1 (0.38) ALDH1A1LMNATP53MAPTTDP1
SCHEMBL8530371 0.85 HINT1 (0.40) ALDH1A1LMNATP53MAPTTDP1
SCHEMBL8530537 0.85 P2RX3 (0.46) ALDH1A1LMNATP53MAPTTDP1
SCHEMBL8530375 0.85 P2RX3 (0.46) ALDH1A1LMNATP53MAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5821236-A Tumor treatment with arabinofuranosyl purine derivatives GLAXO WELLCOME INC. (US) 1998-10-13 US disclosed
US-5747472-A ANTICARCINOGENIC AGENTS AND ANTITUMOR AGENTS GLAXO WELLCOME INC. (US) 1998-05-05 US disclosed
EP-0539479-B1 HETEROCYCLIC COMPOUNDS WELLCOME FOUND (GB) 1997-04-16 EP disclosed
WO-1992001456-A1 HETEROCYCLIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1992-02-06 WO disclosed