SCHEMBL8529909

SCHEMBL8529909

CCOC(=O)c1cn(CCc2ccccc2)nc1N

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 7/20 0.61
ADORA2A P29274 7/20 0.61
ADORA1 P30542 6/20 0.61
ADORA2B P29275 1/20 0.61
TSHR P16473 3/20 0.54
SMN1; SMN2 Q16637 4/20 0.52
MAPT P10636 3/20 0.52
NPC1 O15118 3/20 0.51
RAB9A P51151 3/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
MAPK1 P28482 1/20 0.47
ALDH1A1 P00352 5/20 0.47
HSD17B10 Q99714 1/20 0.47
NFKB1 P19838 1/20 0.46
NFKB2 Q00653 1/20 0.46
RELA Q04206 1/20 0.46
HPGD P15428 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4544356 0.87 ALDH1A1 (0.57) ADORA3ADORA2AADORA1ADORA2BTSHR
SCHEMBL12429197 0.81 TEAD2 (0.45) ADORA3ADORA2AADORA1ADORA2BTSHR
SCHEMBL175330 0.80 ALDH1A1 (0.46) ADORA3ADORA2AADORA1TSHRSMN1; SMN2
SCHEMBL31714887 0.79 TEAD2 (0.43) ADORA3ADORA2AADORA1ADORA2BTSHR
SCHEMBL15884432 0.79 TEAD2 (0.48) ADORA3ADORA2AADORA1ADORA2BTSHR
SCHEMBL2079861 0.76 NPSR1 (0.64) ADORA2AADORA1TSHRSMN1; SMN2MAPT
SCHEMBL645045 0.76 ADORA3 (0.54) ADORA3ADORA2AADORA1TSHRSMN1; SMN2
SCHEMBL31715177 0.76 ALDH1A1 (0.43) ADORA3ADORA2AADORA1TSHRSMN1; SMN2
SCHEMBL17785298 0.76 ALDH1A1 (0.45) ADORA2AADORA1TSHRSMN1; SMN2MAPT
SCHEMBL31352252 0.75 ADORA3 (0.57) ADORA3ADORA2AADORA1TSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5846991-A Pyrazole derivatives NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 1998-12-08 US disclosed
US-5840909-A Pyrazole derivatives NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 1998-11-24 US disclosed
US-5817828-A HYPOTENSIVE AGENTS; CARDIOVASCULAR DISORDERS; VISION DEFECTS NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 1998-10-06 US disclosed
US-5721264-A EXHIBIT ANTAGONISTIC EFFECT AGAINST ANGIOTENSIN II; USEFUL FOR PREVENTION AND REMEDY OF HYPERTENSION, CONGESTIVE HEARTFAILURE, CHRONIC RENAL INSUFFICIENCY, ALDOSTERONISM NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-24 US disclosed
EP-0693480-A1 PYRAZOLE DERIVATIVE NISSAN CHEMICAL INDUSTRIES, LIMITED (JP) 1996-01-24 EP disclosed