SCHEMBL175330

SCHEMBL175330

CCOC(=O)c1cn(CC)nc1N

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
HSD17B10 Q99714 3/20 0.46
CSNK1D P48730 1/20 0.45
TSHR P16473 4/20 0.44
KDM4E B2RXH2 4/20 0.43
RAB9A P51151 4/20 0.43
NPC1 O15118 3/20 0.43
HPGD P15428 2/20 0.43
SMN1; SMN2 Q16637 3/20 0.42
GAA P10253 2/20 0.42
MAPT P10636 2/20 0.42
ALOX15 P16050 1/20 0.42
ATM Q13315 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MAPK1 P28482 1/20 0.42
TEAD2 Q15562 1/20 0.42
TP53 P04637 1/20 0.42
ADORA3 P0DMS8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31715177 0.86 ALDH1A1 (0.43) ALDH1A1MEN1KMT2AHSD17B10CSNK1D
SCHEMBL12429197 0.86 TEAD2 (0.45) ALDH1A1MEN1KMT2AHSD17B10CSNK1D
SCHEMBL31352252 0.85 ADORA3 (0.57) ALDH1A1MEN1KMT2AHSD17B10CSNK1D
SCHEMBL15884432 0.84 TEAD2 (0.48) ALDH1A1MEN1KMT2AHSD17B10CSNK1D
SCHEMBL20098732 0.84 KDM4E (0.45) ALDH1A1MEN1KMT2AHSD17B10CSNK1D
SCHEMBL31714773 0.84 KDM4E (0.48) ALDH1A1MEN1KMT2AHSD17B10CSNK1D
SCHEMBL3809702 0.84 KDM4E (0.42) ALDH1A1MEN1KMT2AHSD17B10CSNK1D
SCHEMBL31714887 0.84 TEAD2 (0.43) ALDH1A1MEN1KMT2AHSD17B10CSNK1D
SCHEMBL23273647 0.83 L3MBTL1 (0.47) ALDH1A1MEN1KMT2AHSD17B10TSHR
SCHEMBL645045 0.83 ADORA3 (0.54) ALDH1A1MEN1KMT2AHSD17B10CSNK1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250333424-A1 ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. 2025-10-30 US disclosed
CN-116096719-A Pyridazinylamino derivatives as ALK5 inhibitors 奇斯药制品公司 2023-05-09 CN disclosed
EP-3324977-B1 BENZODIAZEPINE DERIVATIVES AS RSV INHIBITORS ENANTA PHARM INC (US) 2022-07-13 EP disclosed
US-10881666-B2 Combination pharmaceutical agents as RSV inhibitors ENANTA PHARMACEUTICALS, INC. (US) 2021-01-05 US disclosed
US-10865215-B2 Benzodiazepine derivatives as RSV inhibitors ENANTA PHARMACEUTICALS, INC. (US) 2020-12-15 US disclosed
US-20200223867-A1 BENZODIAZEPINE DERIVATIVES AS RSV INHIBITORS ENANTA PHARM INC (US) 2020-07-16 US disclosed
US-10570153-B2 Benzodiazepine derivatives as RSV inhibitors ENANTA PHARMACEUTICALS, INC. (US) 2020-02-25 US disclosed
US-20190192535-A1 COMBINATION PHARMACEUTICAL AGENTS AS RSV INHIBITORS ENANTA PHARMACEUTICALS, INC. 2019-06-27 US disclosed
US-9957281-B2 Benzodiazepine derivatives as RSV inhibitors ENANTA PHARMACEUTICALS, INC. (US) 2018-05-01 US disclosed
US-20130303533-A1 AZOLOPYRIDINE AND AZOLOPYRIMIDINE COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2013-11-14 US disclosed
WO-2012030924-A1 AZOLOPYRIDINE AND AZOLOPYRIMIDINE COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2012-03-08 WO disclosed
US-7538135-B2 Benzenesulfonylamino compounds and pharmaceutical compositions containing these compounds NOVARTIS AG (CH) 2009-05-26 US disclosed
US-20090062365-A1 Pyrazoles for the Treatment of GERD and IBS ASTRAZENECA AB (SE) 2009-03-05 US disclosed
US-20090062365-A1 Pyrazoles for the Treatment of GERD and IBS ASTRAZENECA AB (SE) 2009-03-05 US disclosed
US-20090062365-A1 Pyrazoles for the Treatment of GERD and IBS ASTRAZENECA AB (SE) 2009-03-05 US disclosed
EP-1966150-A1 PYRAZOLES FOR THE TREATMENT OF GERD AND IBS AstraZeneca AB (SE) 2008-09-10 EP disclosed
WO-2007073297-A1 PYRAZOLES FOR THE TREATMENT OF GERD AND IBS ASTRAZENECA AB (SE) 2007-06-28 WO disclosed
US-20070043020-A1 Benzenesulfonylamino compounds and pharmaceutical compositions containing these compounds NOVARTIS AG (CH) 2007-02-22 US disclosed
EP-1646628-A1 BENZENESULFONYLAMINO COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS Novartis AG (CH) 2006-04-19 EP disclosed
WO-2005005421-A1 BENZENESULFONYLAMINO COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS NOVARTIS AG (CH) 2005-01-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10865215-B2 Benzodiazepine derivatives as RSV inhibitors GABRA5, GABRA1, GABBR2 ALDH1A1 621/4885MEN1 3463/4885KMT2A 1493/4885
US-20090062365-A1 Pyrazoles for the Treatment of GERD and IBS GRPR, GABRB3, GABRB1 ALDH1A1 1412/4885MEN1 4453/4885KMT2A 3841/4885
US-10881666-B2 Combination pharmaceutical agents as RSV inhibitors SERPINB1, FURIN, HIF1AN ALDH1A1 3562/4885MEN1 3503/4885KMT2A 3794/4885
US-20070043020-A1 Benzenesulfonylamino compounds and pharmaceutical compositions containing these compounds PPARG, PPARA, PPARD ALDH1A1 1496/4885MEN1 4484/4885KMT2A 2246/4885
US-10570153-B2 Benzodiazepine derivatives as RSV inhibitors GABRA5, GABRA1, GABBR2 ALDH1A1 621/4885MEN1 3463/4885KMT2A 1493/4885
US-20130303533-A1 AZOLOPYRIDINE AND AZOLOPYRIMIDINE COMPOUNDS AND METHODS OF USE THEREOF JAK3, JAK2, JAK1 ALDH1A1 3689/4885MEN1 2341/4885KMT2A 610/4885
US-20250333424-A1 ANTIVIRAL COMPOUNDS MAVS, EIF2AK2, IRF3 ALDH1A1 3515/4885MEN1 4238/4885KMT2A 4296/4885
US-20200223867-A1 BENZODIAZEPINE DERIVATIVES AS RSV INHIBITORS GABRA5, GABRA1, GABBR2 ALDH1A1 621/4885MEN1 3463/4885KMT2A 1493/4885
US-20190192535-A1 COMBINATION PHARMACEUTICAL AGENTS AS RSV INHIBITORS SERPINB1, FURIN, HIF1AN ALDH1A1 3562/4885MEN1 3503/4885KMT2A 3794/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.