SCHEMBL8529947

SCHEMBL8529947

CCOC(=O)C(CC(C)C)C(CSc1ccc2ccccc2c1)[PH2]=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
CAPN1 P07384 1/20 0.40
CTSB P07858 1/20 0.40
ANPEP P15144 1/20 0.37
EPHX1 P07099 1/20 0.37
KDM4E B2RXH2 3/20 0.36
NPC1 O15118 2/20 0.36
GAA P10253 2/20 0.36
ALDH1A1 P00352 3/20 0.36
CNR2 P34972 1/20 0.35
PLA2G10 O15496 1/20 0.35
CASP1 P29466 1/20 0.35
CASP3 P42574 1/20 0.35
CASP7 P55210 1/20 0.35
CASP6 P55212 1/20 0.35
CASP8 Q14790 1/20 0.35
BACE1 P56817 5/20 0.35
KMT2A Q03164 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8530425 0.87 MTNR1A (0.41) NPC1ALDH1A1KMT2AMAPK1L3MBTL1
SCHEMBL7449784 0.82 PRNP (0.54) CYP2C9KDM4ENPC1GAAALDH1A1
SCHEMBL7050182 0.81 MAPK1 (0.37) KDM4ENPC1ALDH1A1KMT2AMAPK1
SCHEMBL8528289 0.81 CDC25B (0.39) KDM4EALDH1A1CASP1CASP3CASP7
SCHEMBL27041447 0.78 CYP3A4 (0.52) CYP3A4CYP2C9CYP2C19ANPEPEPHX1
SCHEMBL7049697 0.78 L3MBTL1 (0.35) CYP2C9KDM4EGAAALDH1A1KMT2A
SCHEMBL7050114 0.73 CAPN1 (0.38) CYP3A4CYP2C9CYP2C19CAPN1CTSB
SCHEMBL7905195 0.71 EPHX1 (0.65) EPHX1KDM4EGAAALDH1A1KMT2A
SCHEMBL9067733 0.71 CAPN1 (0.44) CYP3A4CYP2C9CYP2C19CAPN1CTSB
SCHEMBL9067046 0.70 SMN1; SMN2 (0.41) ALDH1A1KMT2AMAPTHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5773428-A BONE DISORDERS SYNTEX (U.S.A.) INC. (US) 1998-06-30 US disclosed
EP-0726903-A1 MATRIX METALLOPROTEASE INHIBITORS SYNTEX INC (US) 1996-08-21 EP disclosed
WO-1995012603-A1 MATRIX METALLOPROTEASE INHIBITORS________________________________ SYNTEX (U.S.A.) INC. (US) 1995-05-11 WO disclosed