SCHEMBL8530933

SCHEMBL8530933

Fc1cc(C(Cl)(Cl)Cl)c(F)c(Cl)c1F

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8530898 0.81 ALDH1A1 (0.32) CYP3A4TSHRTDP1
SCHEMBL8525893 0.81 CYP3A4 (0.33) CYP3A4TSHRMAPK1TDP1
SCHEMBL8728803 0.81 TSHR (0.38) CYP3A4TSHRMAPK1TDP1
SCHEMBL6889568 0.80 CYP3A4 (0.31) CYP3A4TSHRMAPK1TDP1
SCHEMBL18167294 0.76 TSHR (0.38) CYP3A4TSHRMAPK1TDP1
SCHEMBL2931707 0.76 CA1 (0.38) CYP3A4
SCHEMBL8974765 0.73 CYP3A4 (0.34) CYP3A4TSHRMAPK1TDP1
SCHEMBL10742911 0.71 EPAS1 (0.33) CYP3A4TSHRTDP1
SCHEMBL8160044 0.71 CYP3A4 (0.43) CYP3A4TSHRMAPK1TDP1
SCHEMBL7057611 0.70 TSHR (0.46) CYP3A4TSHRMAPK1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0725050-B1 Process for the preparation of nuclear halides of benzotrichlorides from the corresponding benzotrifluorides BAYER AG (DE) 1998-12-30 EP disclosed
US-5672791-A Process for the preparation of nuclear-halogenated benzotrichlorides from the corresponding benzotrifluorides BAYER AKTIENGESELLSCHAFT (DE) 1997-09-30 US disclosed
EP-0725050-A1 Process for the preparation of nuclear halides of benzotrichlorides from the corresponding benzotrifluorides BAYER AG (DE) 1996-08-07 EP disclosed