SCHEMBL8533186

SCHEMBL8533186

CCCc1nnnn1-c1ccc(O)c(C=O)c1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CDK1 P06493 1/20 0.38
PTGS2 P35354 2/20 0.38
HSD11B1 P28845 2/20 0.37
ERN1 O75460 5/20 0.37
TP53 P04637 1/20 0.37
MAPT P10636 1/20 0.36
ALPL P05186 1/20 0.36
ALPG P10696 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8532995 0.91 NPC1 (0.42) ALDH1A1LMNANPSR1L3MBTL1CDK1
SCHEMBL8531571 0.82 TACR1 (0.45) ALDH1A1LMNANPSR1L3MBTL1TP53
SCHEMBL3814197 0.80 LMNA (0.47) LMNACDK1ERN1ALPLALPG
SCHEMBL8533644 0.76 SMN1; SMN2 (0.57) ALDH1A1LMNAL3MBTL1ERN1TP53
SCHEMBL8530581 0.76 ALDH1A1 (0.53) ALDH1A1LMNANPSR1L3MBTL1PTGS2
SCHEMBL311546 0.74 ERN1 (0.38) ALDH1A1LMNACDK1ERN1MAPT
SCHEMBL8529476 0.73 TSHR (0.56) ALDH1A1LMNANPSR1L3MBTL1PTGS2
SCHEMBL8529998 0.73 ESR2 (0.40) ERN1TP53MAPT
SCHEMBL4205207 0.73 TACR1 (0.44) ALDH1A1LMNA
SCHEMBL4414691 0.70 HSD11B1 (0.57) ALDH1A1LMNANPSR1L3MBTL1HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5843966-A Piperidine derivatives GLAXO GROUP LIMITED (GB) 1998-12-01 US disclosed
EP-0720609-B1 3-(5-TETRAZOLYL-BENZYL)AMINO-PIPERIDINE DERIVATIVES AND ANTAGONISTS OF TACHYKININS GLAXO GROUP LTD (GB) 1998-11-11 EP disclosed
US-5703240-A ANALGESICS; ANTIINFLAMMATORY AGENTS; NERVOUS SYSTEM DISORDERS; PSYCHOLOGICAL DISORDERS; GASTROINTESTINAL DISORDERS GLAXO GROUP LIMITED (GB) 1997-12-30 US disclosed
EP-0720609-A1 3-(5-TETRAZOLYL-BENZYL)AMINO-PIPERIDINE DERIVATIVES AND ANTAGONISTS OF TACHYKININS GLAXO GROUP LIMITED (GB) 1996-07-10 EP disclosed
WO-1995008549-A1 3-(5-TETRAZOLYL-BENZYL)AMINO-PIPERIDINE DERIVATIVES AND ANTAGONISTS OF TACHYKININS GLAXO GROUP LIMITED (GB) 1995-03-30 WO disclosed