SCHEMBL8533938

SCHEMBL8533938

Cc1cccc(Sc2ccccc2C(=O)N(C)C)c1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.53
MEN1 O00255 3/20 0.53
KMT2A Q03164 3/20 0.53
HPGD P15428 2/20 0.53
MAPT P10636 1/20 0.53
SLC6A4 P31645 1/20 0.44
SIRT1 Q96EB6 1/20 0.44
HTR1A P08908 2/20 0.43
HTR3A P46098 2/20 0.43
ICAM1 P05362 1/20 0.41
SELE P16581 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
KEAP1 Q14145 1/20 0.40
HTT P42858 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
SLC6A9 P48067 2/20 0.38
POLB P06746 1/20 0.38
SCN2A Q99250 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8536289 0.85 MEN1 (0.53) ALDH1A1MEN1KMT2AHPGDMAPT
SCHEMBL11749787 0.84 SIRT1 (0.61) ALDH1A1MEN1KMT2AHPGDMAPT
SCHEMBL8530243 0.83 MEN1 (0.53) ALDH1A1MEN1KMT2AMAPTSIRT1
SCHEMBL8531894 0.82 SIRT1 (0.46) ALDH1A1MEN1KMT2AHPGDMAPT
SCHEMBL5833804 0.82 KMT2A (0.50) ALDH1A1MEN1KMT2AHPGDMAPT
SCHEMBL8533542 0.81 SLC6A4 (0.57) ALDH1A1MEN1KMT2AHPGDMAPT
SCHEMBL8534092 0.81 ALDH1A1 (0.69) ALDH1A1MEN1KMT2AHPGDMAPT
SCHEMBL8530163 0.77 ALDH1A1 (0.54) ALDH1A1MEN1KMT2AHPGDMAPT
SCHEMBL8529733 0.77 MEN1 (0.54) ALDH1A1MEN1KMT2AHPGDMAPT
SCHEMBL8530329 0.73 ALDH1A1 (0.50) ALDH1A1MEN1KMT2AHPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0859757-A1 DERIVATES OF N,N-DIMETHYL-2-(ARYLTHIO)BENZYLAMINE, THEIR SALTS, METHODS OF PREPARATION AND THEIR USE IN PHARMACEUTICAL MEDICAMENTS Farmak A.S. (CZ) 1998-08-26 EP disclosed
WO-1997017325-A1 DERIVATES OF N,N-DIMETHYL-2-(ARYLTHIO)BENZYLAMINE, THEIR SALTS, METHODS OF PREPARATION AND THEIR USE IN PHARMACEUTICAL MEDICAMENTS FARMAK A.S. (CZ) 1997-05-15 WO disclosed
EP-0396827-A1 2-Phenylthiobenzylamine dervivatives and acid addition salts thereof SPOFA Spojené Podniky Pro Zdravotnickou Vyrobu (CS) 1990-11-14 EP disclosed