SCHEMBL8536289

SCHEMBL8536289

CN(C)C(=O)c1cccc(Sc2ccccc2C(=O)N(C)C)c1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.53
KMT2A Q03164 4/20 0.53
ALDH1A1 P00352 3/20 0.53
HPGD P15428 3/20 0.53
MAPT P10636 2/20 0.53
SLC6A4 P31645 1/20 0.44
SIRT1 Q96EB6 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.41
PMM2 O15305 1/20 0.40
MPI P34949 1/20 0.40
PHOSPHO1 Q8TCT1 1/20 0.40
KIF11 P52732 1/20 0.40
LMNA P02545 1/20 0.40
KEAP1 Q14145 1/20 0.40
HTT P42858 1/20 0.40
ERN1 O75460 1/20 0.38
SLC6A9 P48067 3/20 0.38
RARG P13631 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8533938 0.85 ALDH1A1 (0.53) MEN1KMT2AALDH1A1HPGDMAPT
SCHEMBL11749787 0.84 SIRT1 (0.61) MEN1KMT2AALDH1A1HPGDMAPT
SCHEMBL8530163 0.83 ALDH1A1 (0.54) MEN1KMT2AALDH1A1HPGDMAPT
SCHEMBL16495410 0.82 ERN1 (0.50) MEN1KMT2AALDH1A1HPGDMAPT
SCHEMBL5833804 0.82 KMT2A (0.50) MEN1KMT2AALDH1A1HPGDMAPT
SCHEMBL8533542 0.81 SLC6A4 (0.57) MEN1KMT2AALDH1A1HPGDMAPT
SCHEMBL8534092 0.81 ALDH1A1 (0.69) MEN1KMT2AALDH1A1HPGDMAPT
SCHEMBL2480090 0.77 HPGD (0.60) MEN1KMT2AALDH1A1HPGDSMN1; SMN2
SCHEMBL8529733 0.77 MEN1 (0.54) MEN1KMT2AALDH1A1HPGDMAPT
SCHEMBL1447741 0.75 KDM4E (0.59) ALDH1A1HPGDMAPTSIRT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5922914-A REDUCING 2,4-DIHYDRO-6-METHYL-4-PHENYL-2H-BENZOPYRAN-2-ONE WITH A REDUCING AGENT TO FORM 3,4-DIHYDRO-6-METHYL-4-PHENYL-2H-BENZOPYRAN-2-OL CHEMICAL INTERMEDIATE, REDUCTIVELY AMINATING THE HYDROXY COMPOUND PHARMACIA & UPJOHN COMPANY (US) 1999-07-13 US claimed
EP-0859757-A1 DERIVATES OF N,N-DIMETHYL-2-(ARYLTHIO)BENZYLAMINE, THEIR SALTS, METHODS OF PREPARATION AND THEIR USE IN PHARMACEUTICAL MEDICAMENTS Farmak A.S. (CZ) 1998-08-26 EP disclosed
WO-1997017325-A1 DERIVATES OF N,N-DIMETHYL-2-(ARYLTHIO)BENZYLAMINE, THEIR SALTS, METHODS OF PREPARATION AND THEIR USE IN PHARMACEUTICAL MEDICAMENTS FARMAK A.S. (CZ) 1997-05-15 WO disclosed