SCHEMBL8533975

SCHEMBL8533975

O=C(O)c1cc(F)ccc1Sc1ccc(C(F)(F)F)cc1[N+](=O)[O-]

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.58
LMNA P02545 4/20 0.58
HTT P42858 1/20 0.58
AKR1B1 P15121 2/20 0.50
AKR1C4 P17516 2/20 0.50
AKR1C3 P42330 2/20 0.50
AKR1C2 P52895 2/20 0.50
AKR1C1 Q04828 2/20 0.50
MEN1 O00255 4/20 0.49
KMT2A Q03164 4/20 0.49
ALDH1A1 P00352 3/20 0.49
CYP1A2 P05177 1/20 0.49
POLB P06746 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C19 P33261 1/20 0.49
GAA P10253 1/20 0.48
HPGD P15428 1/20 0.48
THRB P10828 2/20 0.45
PDE7A Q13946 1/20 0.45
TTR P02766 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7824348 0.86 MAPT (0.77) MAPTLMNAHTTAKR1B1AKR1C4
SCHEMBL4436473 0.86 MPO (0.50) MAPTLMNAHTTMEN1KMT2A
SCHEMBL4637151 0.84 APEX1 (0.54) MAPTLMNAMEN1KMT2AALDH1A1
SCHEMBL8530063 0.80 ALDH1A1 (0.57) MAPTLMNAHTTMEN1KMT2A
SCHEMBL1645800 0.80 MAPT (0.60) MAPTLMNAHTTMEN1KMT2A
SCHEMBL15911983 0.78 ALDH1A1 (0.56) MAPTLMNAHTTAKR1B1AKR1C4
SCHEMBL8535062 0.78 KCNK2 (0.46) MAPTLMNAHTTALDH1A1CYP1A2
SCHEMBL4433443 0.78 ALDH1A1 (0.52) MAPTHTTMEN1KMT2AALDH1A1
SCHEMBL442397 0.77 HPD (0.60) MAPTLMNAHTTAKR1B1AKR1C4
SCHEMBL4448254 0.77 CFTR (0.49) ALDH1A1CYP2C19HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0859757-A1 DERIVATES OF N,N-DIMETHYL-2-(ARYLTHIO)BENZYLAMINE, THEIR SALTS, METHODS OF PREPARATION AND THEIR USE IN PHARMACEUTICAL MEDICAMENTS Farmak A.S. (CZ) 1998-08-26 EP disclosed
WO-1997017325-A1 DERIVATES OF N,N-DIMETHYL-2-(ARYLTHIO)BENZYLAMINE, THEIR SALTS, METHODS OF PREPARATION AND THEIR USE IN PHARMACEUTICAL MEDICAMENTS FARMAK A.S. (CZ) 1997-05-15 WO disclosed