SCHEMBL8533982

SCHEMBL8533982

COc1ccc(N(C(=O)c2ccccc2)c2ccccc2)cc1NC(=S)Nc1cc(Cl)cc(Cl)c1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 10/20 0.53
ALDH1A1 P00352 8/20 0.53
MEN1 O00255 8/20 0.53
MAPT P10636 6/20 0.53
GAA P10253 5/20 0.53
LMNA P02545 2/20 0.50
HPGD P15428 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.47
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2C19 P33261 2/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
XBP1 P17861 1/20 0.45
HTT P42858 1/20 0.45
KDM4E B2RXH2 1/20 0.44
POLB P06746 1/20 0.42
SMO Q99835 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6812705 0.80 ALDH1A1 (0.60) KMT2AALDH1A1MEN1MAPTGAA
SCHEMBL8533988 0.79 NR3C2 (0.40) KMT2AALDH1A1MEN1MAPTGAA
SCHEMBL6813184 0.78 ALDH1A1 (0.57) KMT2AALDH1A1MEN1MAPTGAA
SCHEMBL6812366 0.77 KMT2A (0.58) KMT2AALDH1A1MEN1MAPTGAA
SCHEMBL6813779 0.74 MEN1 (0.55) KMT2AALDH1A1MEN1MAPTGAA
SCHEMBL6809706 0.72 HDAC8 (0.60) KMT2AALDH1A1MEN1MAPTGAA
SCHEMBL6812397 0.72 ALDH1A1 (0.57) KMT2AALDH1A1MEN1MAPTGAA
SCHEMBL5450034 0.72 GAA (0.76) KMT2AALDH1A1MEN1MAPTGAA
SCHEMBL6813268 0.71 HDAC8 (0.56) KMT2AALDH1A1MEN1MAPTGAA
SCHEMBL6813288 0.71 ALDH1A1 (0.65) KMT2AALDH1A1MEN1MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042276-A1 THIOUREA COMPOUNDS, COMPOSITIONS AND METHODS OF TREATING OR PREVENTING INFLAMMATORY DISEASES AND ATHEROSCLEROSIS WARNER-LAMBERT COMPANY LLC (US) 2000-10-11 EP disclosed
WO-1999032433-A1 THIOUREA AND BENZAMIDE COMPOUNDS, COMPOSITIONS AND METHODS OF TREATING OR PREVENTING INFLAMMATORY DISEASES AND ATHEROSCLEROSIS WARNER-LAMBERT COMPANY (US) 1999-07-01 WO disclosed