SCHEMBL8534863

SCHEMBL8534863

CC(C)[C@H](N)C(=O)N(C(=O)[C@@H](NC(=O)CCCCCNC(=O)OCc1ccccc1)C(C)C)C(Cc1ccccc1)C(O)C(Cc1ccccc1)N(C(=O)[C@@H](N)C(C)C)C(=O)[C@@H](NC(=O)CCCCC(=O)O)C(C)C

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.47
FOLH1 Q04609 7/20 0.43
PTGER4 P35408 3/20 0.42
SIRT2 Q8IXJ6 1/20 0.40
CTSL P07711 1/20 0.40
CTSB P07858 1/20 0.40
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
TGM2 P21980 1/20 0.39
CPB1 P15086 1/20 0.39
CPB2 Q96IY4 1/20 0.39
CAPN1 P07384 1/20 0.39
CAPN2 P17655 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8539753 0.94 CTSD (0.39) HTTFOLH1SIRT2CTSLCTSB
SCHEMBL8534831 0.88 HTT (0.46) HTTFOLH1PTGER4
SCHEMBL8536372 0.86 MMP2 (0.46) CPB2
SCHEMBL7279640 0.83 HTT (0.41) HTTFOLH1PTGER4SIRT2CPB1
SCHEMBL8539750 0.82 CTSD (0.42) HTTFOLH1CTSLCTSBCTSS
SCHEMBL7279627 0.81 PTGER4 (0.41) HTTFOLH1PTGER4
SCHEMBL8534869 0.80 CTSD (0.58) HTTFOLH1PTGER4
SCHEMBL6443882 0.78 HTT (0.56) HTTFOLH1SIRT2TGM2CPB1
SCHEMBL6443877 0.78 HTT (0.56) HTTFOLH1SIRT2TGM2CPB1
SCHEMBL9741444 0.77 CTSD (0.37) FOLH1SIRT2CPB1CPB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
US-5142056-A Human immunodeficiency virus protease inhibitor ABBOTT LABORATORIES (US) 1992-08-25 US disclosed