SCHEMBL8539753

SCHEMBL8539753

COC(=O)CCCCC(=O)N[C@H](C(=O)N(C(=O)[C@@H](N)C(C)C)C(Cc1ccccc1)C(O)C(Cc1ccccc1)N(C(=O)[C@@H](N)C(C)C)C(=O)[C@@H](NC(=O)CCCCCNC(=O)OCc1ccccc1)C(C)C)C(C)C

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSD P07339 1/20 0.39
HTT P42858 1/20 0.39
BACE1 P56817 1/20 0.39
SIRT2 Q8IXJ6 2/20 0.39
CTSL P07711 1/20 0.39
CTSB P07858 1/20 0.39
CTSS P25774 1/20 0.39
CTSK P43235 1/20 0.39
REN P00797 1/20 0.39
CPB1 P15086 1/20 0.38
CPB2 Q96IY4 1/20 0.38
TGM2 P21980 1/20 0.38
FOLH1 Q04609 2/20 0.38
SIRT1 Q96EB6 1/20 0.38
SIRT3 Q9NTG7 1/20 0.38
CAPN1 P07384 1/20 0.38
CAPN2 P17655 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8534863 0.94 HTT (0.47) HTTSIRT2CTSLCTSBCTSS
SCHEMBL8539750 0.89 CTSD (0.42) CTSDHTTBACE1CTSLCTSB
SCHEMBL9741444 0.83 CTSD (0.37) CTSDBACE1SIRT2RENCPB1
SCHEMBL8534831 0.82 HTT (0.46) CTSDHTTFOLH1
SCHEMBL8539759 0.81 CTSD (0.57) CTSDREN
SCHEMBL8536372 0.80 MMP2 (0.46) CTSDCPB2
SCHEMBL7279640 0.78 HTT (0.41) HTTSIRT2CPB1CPB2FOLH1
SCHEMBL6443882 0.77 HTT (0.56) HTTSIRT2CPB1CPB2TGM2
SCHEMBL6443877 0.77 HTT (0.56) HTTSIRT2CPB1CPB2TGM2
SCHEMBL6447440 0.76 HTT (0.57) HTTSIRT2CPB1CPB2TGM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed