SCHEMBL8535449

SCHEMBL8535449

Cc1ncc(CCNC(=O)C2CCCN(CC(c3ccccc3)c3ccccc3)C2)n1Cc1ccc(C#N)cc1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 10/20 0.48
FNTA P49354 3/20 0.47
FNTB P49356 3/20 0.47
PGGT1B P53609 3/20 0.47
CHRM4 P08173 2/20 0.44
ERG P11308 3/20 0.43
CYP3A4 P08684 1/20 0.42
TP53 P04637 1/20 0.42
POLB P06746 1/20 0.42
MAPT P10636 1/20 0.42
CHRM2 P08172 1/20 0.42
CHRM5 P08912 1/20 0.42
CHRM1 P11229 1/20 0.42
CYP2C9 P11712 1/20 0.42
CCR2 P41597 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8097241 1.00 GPBAR1 (0.48) GPBAR1FNTAFNTBPGGT1BCHRM4
SCHEMBL8097422 0.89 GPBAR1 (0.49) GPBAR1FNTAFNTBPGGT1BCHRM4
SCHEMBL8434674 0.89 GPBAR1 (0.49) GPBAR1FNTAFNTBPGGT1BCHRM4
SCHEMBL446562 0.85 FNTA (0.54) FNTAFNTBPGGT1B
SCHEMBL8097236 0.85 CCR5 (0.44) GPBAR1FNTAFNTBPGGT1BCHRM4
SCHEMBL8534261 0.82 FNTA (0.48) GPBAR1FNTAFNTBPGGT1BTP53
SCHEMBL8095893 0.82 FNTA (0.48) GPBAR1FNTAFNTBPGGT1BTP53
SCHEMBL8433745 0.82 FNTA (0.51) FNTAFNTBPGGT1B
SCHEMBL8095475 0.82 FNTA (0.51) FNTAFNTBPGGT1B
SCHEMBL8444571 0.80 FNTA (0.45) FNTAFNTBPGGT1BCCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5817678-A IMIDAZOLE-CONTAINING PIPERIDINE DERIVATIVES, PEPTIDEMIMETIC MERCK & CO., INC. (US) 1998-10-06 US disclosed